FAIRMol

Z1157836593

Pose ID 2462 Compound 32 Pose 2462

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing
T02
Dihydrofolate reductase Homo sapiens
Ligand Z1157836593
PDB5SD8

3D complex viewer

Strict H-bonds Permissive H-bonds
Viewer legend
Protein receptor
Pocket residues
Cofactor context
Docked ligand
Overall assessment
Reject No SASA yet
Promising but geometrically suspicious
Binding strong Geometry low Native strong SASA missing
Strain ΔE
28.0 kcal/mol
Protein clashes
7
Internal clashes
9
Native overlap
contact recall 0.81, Jaccard 0.81, H-bond role recall 0.00
Burial
100%
Reason: 9 internal clashes
7 protein-contact clashes 9 intramolecular clashes
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.917 kcal/mol/HA) ✓ Good fit quality (FQ -8.22) ✗ High strain energy (28.0 kcal/mol) ✗ No H-bonds detected ✗ Geometry warnings ✗ Protein-contact clashes (7) ✗ Internal clashes (9) ℹ SASA not computed
Score
-22.012
kcal/mol
LE
-0.917
kcal/mol/HA
Fit Quality
-8.22
FQ (Leeson)
HAC
24
heavy atoms
MW
401
Da
LogP
4.84
cLogP
Strain ΔE
28.0 kcal/mol
SASA buried
computing…

Interaction summary

HB 0 HY 24 PI 1 CLASH 0
Final rank4.035Score-22.012
Inter norm-1.046Intra norm0.129
Top1000noExcludedno
Contacts17H-bonds0
Artifact reasongeometry warning; 9 clashes; 7 protein contact clashes; high strain Δ 28.0
Residues
ALA10 ASN65 ASP22 GLY21 ILE61 ILE8 LEU23 LEU68 NAP201 PHE32 PHE35 PRO62 SER60 THR57 TYR122 VAL116 VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Receptor context

1 kept / 0 excluded
Receptor context filtering: interactions and SASA are computed against protein atoms plus allowed cofactors/ions. Native ligand-like HETATM partners are excluded from scoring.
Kept context 1 Excluded HETATM 0
Kept cofactors / ions
A:NAP201

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseHB0
IFP residues
ALA10 ASN65 ASP22 GLN36 GLU31 GLY117 GLY21 ILE61 ILE8 LEU23 LEU68 NAP201 PHE32 PHE35 PRO62 SER60 THR137 THR57 TYR122 VAL116 VAL9
Current overlap17Native recall0.81
Jaccard0.81RMSD-
HB strict0Strict recall0.00
HB same residue+role0HB role recall0.00
HB same residue0HB residue recall0.00

HB · H-bonds

No hb · h-bonds detected for this pose.

PI · π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

HY · Hydrophobic contacts

CLASH · Clashes

No clash · clashes detected for this pose.

All stored poses for this docking hit

PoseFinal rankInter normScoreHBCTCT overlapCT recallHB role rec.RMSDExcluded
2463 2.7987022811904225 -1.08262 -20.9198 0 17 17 0.81 0.00 - no Open
969 2.808571801991689 -1.22264 -25.5784 3 14 0 0.00 0.00 - no Open
2464 2.866885825158193 -1.03673 -21.2526 0 17 17 0.81 0.00 - no Open
970 2.92618531156925 -1.16681 -26.2906 3 14 0 0.00 0.00 - no Open
1220 3.473207146863788 -1.28279 -26.8387 1 14 0 0.00 0.00 - no Open
1221 3.5298908329704504 -1.12772 -25.0807 3 13 0 0.00 0.00 - no Open
2462 4.03491069258468 -1.04639 -22.0124 0 17 17 0.81 0.00 - no Current
2461 4.0643568591372174 -1.03047 -21.4763 1 17 17 0.81 0.20 - no Open
956 4.838840042093441 -0.999945 -19.8731 0 14 0 0.00 0.00 - no Open
1064 5.0312206236412935 -0.973313 -20.1998 1 16 0 0.00 0.00 - no Open
1065 4.8478327579821805 -1.0358 -20.9894 1 16 0 0.00 0.00 - yes Open
1063 5.307139313163413 -0.855698 -17.0141 0 15 0 0.00 0.00 - yes Open
957 5.687680835199031 -0.685719 -13.2604 1 10 0 0.00 0.00 - yes Open
954 7.13543081556128 -1.20858 -26.4233 2 13 0 0.00 0.00 - yes Open
1062 7.9428998618738715 -1.04639 -23.5646 2 15 0 0.00 0.00 - yes Open
955 8.38934841134014 -1.01248 -23.4793 2 12 0 0.00 0.00 - yes Open

Molecular metrics

RDKit SASA burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.012kcal/mol
Ligand efficiency (LE) -0.9172kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -8.220
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 24HA

Physicochemical properties

Molecular weight 401.3Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.84
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 28.04kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 80.27kcal/mol
Minimised FF energy 52.23kcal/mol

SASA & burial

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate SASA burial metrics without blocking the page.