FAIRMol

Z1157836593

Pose ID 14074 Compound 32 Pose 1221

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-1.045 kcal/mol/HA) ✓ Good fit quality (FQ -9.37) ✓ Good H-bonds (3 bonds) ✗ High strain energy (17.0 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-25.081
kcal/mol
LE
-1.045
kcal/mol/HA
Fit Quality
-9.37
FQ (Leeson)
HAC
24
heavy atoms
MW
401
Da
LogP
4.84
cLogP
Strain ΔE
17.0 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 24 π–π 4 Clashes 7 Severe clashes 0
Final rank3.5298908329704504Score-25.0807
Inter norm-1.12772Intra norm0.0826876
Top1000noExcludedno
Contacts13H-bonds3
Artifact reasongeometry warning; 10 clashes; 7 protein contact clashes; moderate strain Δ 17.0
ResiduesA:ARG14;A:ASP161;A:CYS168;A:LEU209;A:MET213;A:NAP301;A:PHE171;A:PHE97;A:PRO210;A:PRO99;A:TRP221;A:TYR174;A:VAL206

Protein summary

258 residues
Protein targetT08Atoms3881
Residues258Chains2
Residue summaryLEU:437; VAL:433; ALA:361; ARG:288; ILE:266; GLU:210; LYS:198; SER:198; ASN:182; THR:154; GLN:153; PHE:140; PRO:140; TYR:126; GLY:112; HIS:103

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
NameTbPTR1_cW_6RX6_ReadyContacts19
PoseOpen native poseH-bonds6
IFP residuesA:ARG14; A:ASP161; A:CYS168; A:GLY205; A:LEU208; A:LEU209; A:LYS178; A:MET213; A:NAP301; A:PHE171; A:PHE97; A:PRO210; A:PRO99; A:SER207; A:SER95; A:TRP221; A:TYR174; A:TYR98; A:VAL206
Current overlap13Native recall0.68
Jaccard0.68RMSD-
H-bond strict1Strict recall0.17
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2463 2.7987022811904225 -1.08262 -20.9198 0 17 0 0.00 0.00 - no Open
969 2.808571801991689 -1.22264 -25.5784 3 14 14 0.74 0.20 - no Open
2464 2.866885825158193 -1.03673 -21.2526 0 17 0 0.00 0.00 - no Open
970 2.92618531156925 -1.16681 -26.2906 3 14 14 0.74 0.20 - no Open
1220 3.473207146863788 -1.28279 -26.8387 1 14 14 0.74 0.00 - no Open
1221 3.5298908329704504 -1.12772 -25.0807 3 13 13 0.68 0.20 - no Current
2462 4.03491069258468 -1.04639 -22.0124 0 17 0 0.00 0.00 - no Open
2461 4.0643568591372174 -1.03047 -21.4763 1 17 0 0.00 0.00 - no Open
956 4.838840042093441 -0.999945 -19.8731 0 14 0 0.00 0.00 - no Open
1064 5.0312206236412935 -0.973313 -20.1998 1 16 0 0.00 0.00 - no Open
1065 4.8478327579821805 -1.0358 -20.9894 1 16 0 0.00 0.00 - yes Open
1063 5.307139313163413 -0.855698 -17.0141 0 15 0 0.00 0.00 - yes Open
957 5.687680835199031 -0.685719 -13.2604 1 10 0 0.00 0.00 - yes Open
954 7.13543081556128 -1.20858 -26.4233 2 13 0 0.00 0.00 - yes Open
1062 7.9428998618738715 -1.04639 -23.5646 2 15 0 0.00 0.00 - yes Open
955 8.38934841134014 -1.01248 -23.4793 2 12 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -25.081kcal/mol
Ligand efficiency (LE) -1.0450kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -9.365
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 24HA

Physicochemical properties

Molecular weight 401.3Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.84
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 17.02kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 124.25kcal/mol
Minimised FF energy 107.23kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.