FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 8 best compound-target hits listed 8 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T03T08T09T14T17T18T21
Z29294093
[H]N([H])/C(O)=C1\C=C(c2ccccc2)S\C1=N/C(=O)Cc1ccc(S(=O)(=O)N2CCOCC2)s1
0.913 0.855 5 0.82 0.87 0.85 0.82 0.91
Z29294093
[H]N([H])C(=O)c1cc(-c2ccccc2)sc1N([H])C(=O)Cc1ccc(S(=O)(=O)N2CCOCC2)s1
0.852 0.815 3 0.85 0.80 0.79

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z29294093
[H]N([H])/C(O)=C1\C=C(c2ccccc2)S\C1=N/C(=O)Cc1ccc(S(=O)(=O)N2CCOCC2)s1
T21
native IFP available
T21
selection_import_t21
0.913 1.000 0.750 native_similarity final_rank_score -46.8966 -0.786972 18 11 Pose
Z29294093
[H]N([H])/C(O)=C1\C=C(c2ccccc2)S\C1=N/C(=O)Cc1ccc(S(=O)(=O)N2CCOCC2)s1
T03
native IFP available
T03
selection_import_t03
0.868 1.000 0.624 native_similarity final_rank_score -49.0529 -0.884942 19 4 Pose
Z29294093
[H]N([H])C(=O)c1cc(-c2ccccc2)sc1N([H])C(=O)Cc1ccc(S(=O)(=O)N2CCOCC2)s1
T08
native IFP available
T08
selection_import_t08
0.852 1.000 0.578 native_similarity final_rank_score -29.8272 -0.995577 14 10 Pose
Z29294093
[H]N([H])/C(O)=C1\C=C(c2ccccc2)S\C1=N/C(=O)Cc1ccc(S(=O)(=O)N2CCOCC2)s1
T09
native IFP available
T09
selection_import_t09
0.852 1.000 0.576 native_similarity final_rank_score -46.3282 -0.793129 20 4 Pose
Z29294093
[H]N([H])/C(O)=C1\C=C(c2ccccc2)S\C1=N/C(=O)Cc1ccc(S(=O)(=O)N2CCOCC2)s1
T01
native IFP available
T01
selection_import_t01
0.822 1.000 0.491 native_similarity final_rank_score -31.1479 -0.821422 15 4 Pose
Z29294093
[H]N([H])/C(O)=C1\C=C(c2ccccc2)S\C1=N/C(=O)Cc1ccc(S(=O)(=O)N2CCOCC2)s1
T14
native IFP available
T14
selection_import_t14
0.819 1.000 0.482 native_similarity final_rank_score -47.0997 -0.732381 13 5 Pose
Z29294093
[H]N([H])C(=O)c1cc(-c2ccccc2)sc1N([H])C(=O)Cc1ccc(S(=O)(=O)N2CCOCC2)s1
T17
native IFP available
T17
selection_import_t17
0.799 1.000 0.425 native_similarity final_rank_score -22.0319 -0.706171 15 8 Pose
Z29294093
[H]N([H])C(=O)c1cc(-c2ccccc2)sc1N([H])C(=O)Cc1ccc(S(=O)(=O)N2CCOCC2)s1
T18
native IFP available
T18
selection_import_t18
0.793 1.000 0.408 native_similarity final_rank_score -24.7022 -0.754114 14 5 Pose