FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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2 compounds in matrix 9 best compound-target hits listed 9 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T03T08T10T14T16T18T19T20
Z49638306
[H]Oc1ccc(/C(C)=N\N([H])C(=O)c2cc(-c3cccnc3)nc3ccccc23)c(O)c1
0.904 0.823 4 0.75 0.84 0.90 0.80
Z49638306
[H]Oc1ccc(/C(C)=N/N([H])C(=O)c2cc(-c3cccnc3)nc3ccccc23)c(O)c1
0.894 0.792 5 0.78 0.79 0.76 0.74 0.89

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z49638306
[H]Oc1ccc(/C(C)=N\N([H])C(=O)c2cc(-c3cccnc3)nc3ccccc23)c(O)c1
T10
native IFP available
T10
dockmulti_91311c650f2e_T10
0.904 1.000 0.727 native_similarity final_rank_score -20.6491 -0.629821 15 5 Pose
Z49638306
[H]Oc1ccc(/C(C)=N/N([H])C(=O)c2cc(-c3cccnc3)nc3ccccc23)c(O)c1
T20
native IFP available
T20
dockmulti_91311c650f2e_T20
0.894 1.000 0.696 native_similarity final_rank_score -25.3759 -0.756591 12 10 Pose
Z49638306
[H]Oc1ccc(/C(C)=N\N([H])C(=O)c2cc(-c3cccnc3)nc3ccccc23)c(O)c1
T08
native IFP available
T08
dockmulti_91311c650f2e_T08
0.844 1.000 0.554 native_similarity final_rank_score -37.7354 -1.21986 14 9 Pose
Z49638306
[H]Oc1ccc(/C(C)=N\N([H])C(=O)c2cc(-c3cccnc3)nc3ccccc23)c(O)c1
T18
native IFP available
T18
dockmulti_91311c650f2e_T18
0.797 1.000 0.419 native_similarity final_rank_score -19.4954 -0.565681 13 6 Pose
Z49638306
[H]Oc1ccc(/C(C)=N/N([H])C(=O)c2cc(-c3cccnc3)nc3ccccc23)c(O)c1
T14
native IFP available
T14
dockmulti_91311c650f2e_T14
0.790 1.000 0.400 native_similarity final_rank_score -26.3523 -0.780324 13 4 Pose
Z49638306
[H]Oc1ccc(/C(C)=N/N([H])C(=O)c2cc(-c3cccnc3)nc3ccccc23)c(O)c1
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.776 1.000 0.360 native_similarity final_rank_score -21.8826 -0.686348 14 6 Pose
Z49638306
[H]Oc1ccc(/C(C)=N/N([H])C(=O)c2cc(-c3cccnc3)nc3ccccc23)c(O)c1
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.760 1.000 0.315 native_similarity final_rank_score -27.8134 -0.775798 15 6 Pose
Z49638306
[H]Oc1ccc(/C(C)=N\N([H])C(=O)c2cc(-c3cccnc3)nc3ccccc23)c(O)c1
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.749 1.000 0.282 native_similarity final_rank_score -26.671 -0.84258 11 9 Pose
Z49638306
[H]Oc1ccc(/C(C)=N/N([H])C(=O)c2cc(-c3cccnc3)nc3ccccc23)c(O)c1
T19
native IFP available
T19
dockmulti_91311c650f2e_T19
0.739 1.000 0.255 native_similarity final_rank_score -28.0721 -0.913857 19 8 Pose