FAIRMol

Z49638306

Pose ID 19359 Compound 667 Pose 1553

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.688 kcal/mol/HA) ✓ Good fit quality (FQ -6.64) ✓ Good H-bonds (5 bonds) ✗ High strain energy (11.8 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-20.649
kcal/mol
LE
-0.688
kcal/mol/HA
Fit Quality
-6.64
FQ (Leeson)
HAC
30
heavy atoms
MW
398
Da
LogP
3.86
cLogP
Strain ΔE
11.8 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 5 Hydrophobic 11 π–π 2 Clashes 15 Severe clashes 0 ⚠ Hydrophobic exposure 39%
⚠️Partial hydrophobic solvent exposure
39% of hydrophobic surface appears solvent-exposed (9/23 atoms). Partial exposure is common but may limit selectivity and membrane permeability.
Non-polar atoms 23 Buried (contacted) 14 Exposed 9 LogP 3.86 H-bonds 5
Exposed fragments: phenyl (6/6 atoms exposed)aliphatic chain/group (3 atoms exposed)
Final rank7.366388362828268Score-20.6491
Inter norm-0.629821Intra norm-0.0584822
Top1000noExcludedno
Contacts15H-bonds5
Artifact reasongeometry warning; 16 clashes; 15 protein contact clashes; moderate strain Δ 15.3
ResiduesA:ARG116;A:ARG140;A:ARG144;A:ASN106;A:ASP13;A:CYS72;A:GLY73;A:GLY75;A:GLY77;A:HIS105;A:HIS14;A:HIS141;A:LEU101;A:THR74;A:TYR49

Protein summary

155 residues
Protein targetT10Atoms4590
Residues155Chains1
Residue summaryILE:494; ARG:384; ALA:360; VAL:352; LEU:304; GLU:300; THR:280; MET:272; LYS:220; ASP:216; TYR:210; HIS:204; GLY:182; SER:176; GLN:170; ASN:140

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name6FXWContacts17
PoseOpen native poseH-bonds16
IFP residuesA:ALA15; A:ARG116; A:ARG140; A:ARG144; A:ASN106; A:ASP13; A:CYS72; A:GLY73; A:GLY75; A:GLY77; A:HIS105; A:HIS14; A:HIS141; A:ILE76; A:LEU101; A:THR74; A:TYR49
Current overlap15Native recall0.88
Jaccard0.88RMSD-
H-bond strict3Strict recall0.23
H-bond same residue+role4Role recall0.36
H-bond same residue4Residue recall0.36

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1906 4.079634371228655 -0.565681 -19.4954 6 13 0 0.00 0.00 - no Open
1904 4.708431710135203 -0.593572 -18.3879 3 8 0 0.00 0.00 - no Open
2552 5.837738885508001 -0.84258 -26.671 9 11 0 0.00 0.00 - no Open
1374 6.9491310065977725 -1.21986 -37.7354 9 14 0 0.00 0.00 - no Open
1553 7.366388362828268 -0.629821 -20.6491 5 15 15 0.88 0.36 - no Current
1549 8.450095171648368 -0.721285 -24.1068 7 16 14 0.82 0.64 - no Open
1900 6.1831904129384965 -0.71915 -21.2671 8 15 0 0.00 0.00 - yes Open
2548 6.398582763603283 -1.07455 -32.5822 7 12 0 0.00 0.00 - yes Open
2553 6.594207675159006 -0.943559 -27.8785 4 14 0 0.00 0.00 - yes Open
2550 6.798936814767271 -0.774692 -22.9352 6 10 0 0.00 0.00 - yes Open
2549 6.971189554398788 -0.915938 -25.9224 4 14 0 0.00 0.00 - yes Open
1905 7.018537068616989 -0.62468 -21.7228 5 9 0 0.00 0.00 - yes Open
2551 7.033853904040928 -0.845777 -26.335 4 15 0 0.00 0.00 - yes Open
1903 7.414535980267811 -0.629732 -20.3929 5 13 0 0.00 0.00 - yes Open
1901 7.816321035401791 -0.673946 -21.3884 4 13 0 0.00 0.00 - yes Open
1548 8.866106778944213 -0.923782 -27.0501 11 19 17 1.00 0.64 - yes Open
1554 9.058924025034537 -0.757065 -21.7722 11 18 16 0.94 0.45 - yes Open
1902 9.330708255049892 -0.712915 -24.4361 3 13 0 0.00 0.00 - yes Open
1907 9.607718702921597 -0.633204 -22.1142 5 14 0 0.00 0.00 - yes Open
1547 9.80770316554089 -0.668429 -17.3057 5 16 14 0.82 0.27 - yes Open
1552 10.005670834294907 -0.777192 -26.0641 9 19 15 0.88 0.36 - yes Open
1550 10.24519874536975 -1.07037 -31.267 12 18 16 0.94 0.45 - yes Open
1375 10.697110617251491 -1.12097 -37.0518 10 19 0 0.00 0.00 - yes Open
1551 11.621956666465433 -0.756254 -18.4723 7 15 13 0.76 0.36 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -20.649kcal/mol
Ligand efficiency (LE) -0.6883kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.640
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 30HA

Physicochemical properties

Molecular weight 398.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.86
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 11.76kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 104.55kcal/mol
Minimised FF energy 92.80kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.