FAIRMol

Z19455379

Pose ID 9721 Compound 1114 Pose 1142

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.711 kcal/mol/HA) ✓ Good fit quality (FQ -6.37) ✓ Good H-bonds (3 bonds) ✗ Very high strain energy (21.0 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-17.057
kcal/mol
LE
-0.711
kcal/mol/HA
Fit Quality
-6.37
FQ (Leeson)
HAC
24
heavy atoms
MW
344
Da
LogP
1.88
cLogP
Strain ΔE
21.0 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 21.0 kcal/mol

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 24 π–π 3 Clashes 9 Severe clashes 0
Final rank3.6340295063126695Score-17.0567
Inter norm-0.862014Intra norm0.133034
Top1000noExcludedno
Contacts18H-bonds3
Artifact reasongeometry warning; 5 clashes; 9 protein contact clashes; high strain Δ 20.2
ResiduesA:ALA34;A:ARG100;A:ARG59;A:ASP54;A:GLN56;A:ILE160;A:ILE47;A:LEU90;A:LEU97;A:MET55;A:NDP301;A:PHE58;A:PHE94;A:PRO91;A:THR184;A:TYR166;A:VAL32;A:VAL33

Protein summary

223 residues
Protein targetT06Atoms3452
Residues223Chains1
Residue summaryARG:408; VAL:352; LYS:308; LEU:304; PRO:238; ILE:209; GLU:195; THR:182; SER:176; ALA:160; PHE:140; ASN:126; GLY:126; ASP:108; GLN:85; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name8RHTContacts21
PoseOpen native poseH-bonds6
IFP residuesA:ALA34; A:ASP54; A:HIS182; A:ILE160; A:ILE47; A:LEU90; A:LEU97; A:MET55; A:NDP301; A:PHE233; A:PHE58; A:PHE94; A:PRO91; A:SER89; A:THR184; A:THR86; A:TRP49; A:TYR166; A:TYR57; A:VAL32; A:VAL33
Current overlap15Native recall0.71
Jaccard0.62RMSD-
H-bond strict2Strict recall0.40
H-bond same residue+role2Role recall0.50
H-bond same residue3Residue recall0.75

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1142 3.6340295063126695 -0.862014 -17.0567 3 18 15 0.71 0.50 - no Current
1141 4.856746952818134 -1.01234 -20.2213 5 18 16 0.76 0.25 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -17.057kcal/mol
Ligand efficiency (LE) -0.7107kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.369
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 24HA

Physicochemical properties

Molecular weight 344.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.88
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 20.99kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 32.35kcal/mol
Minimised FF energy 11.36kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.