FAIRMol

Z19455379

Pose ID 9720 Compound 1114 Pose 1141

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.843 kcal/mol/HA) ✓ Good fit quality (FQ -7.55) ✓ Good H-bonds (5 bonds) ✗ High strain energy (15.8 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-20.221
kcal/mol
LE
-0.843
kcal/mol/HA
Fit Quality
-7.55
FQ (Leeson)
HAC
24
heavy atoms
MW
344
Da
LogP
1.88
cLogP
Strain ΔE
15.8 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 15.8 kcal/mol

Interaction summary

Collapsible panels
H-bonds 5 Hydrophobic 24 π–π 1 Clashes 9 Severe clashes 1
Final rank4.856746952818134Score-20.2213
Inter norm-1.01234Intra norm0.169789
Top1000noExcludedyes
Contacts18H-bonds5
Artifact reasonexcluded; geometry warning; 5 clashes; 1 protein clash; moderate strain Δ 16.0
ResiduesA:ALA34;A:ARG100;A:ARG59;A:ASP54;A:ILE160;A:ILE47;A:LEU90;A:LEU97;A:MET55;A:NDP301;A:PHE58;A:PHE94;A:PRO91;A:THR184;A:TYR166;A:TYR57;A:VAL32;A:VAL33

Protein summary

223 residues
Protein targetT06Atoms3452
Residues223Chains1
Residue summaryARG:408; VAL:352; LYS:308; LEU:304; PRO:238; ILE:209; GLU:195; THR:182; SER:176; ALA:160; PHE:140; ASN:126; GLY:126; ASP:108; GLN:85; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name8RHTContacts21
PoseOpen native poseH-bonds6
IFP residuesA:ALA34; A:ASP54; A:HIS182; A:ILE160; A:ILE47; A:LEU90; A:LEU97; A:MET55; A:NDP301; A:PHE233; A:PHE58; A:PHE94; A:PRO91; A:SER89; A:THR184; A:THR86; A:TRP49; A:TYR166; A:TYR57; A:VAL32; A:VAL33
Current overlap16Native recall0.76
Jaccard0.70RMSD-
H-bond strict1Strict recall0.20
H-bond same residue+role1Role recall0.25
H-bond same residue2Residue recall0.50

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1142 3.6340295063126695 -0.862014 -17.0567 3 18 15 0.71 0.50 - no Open
1141 4.856746952818134 -1.01234 -20.2213 5 18 16 0.76 0.25 - yes Current

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -20.221kcal/mol
Ligand efficiency (LE) -0.8426kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.551
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 24HA

Physicochemical properties

Molecular weight 344.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.88
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 15.84kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 29.08kcal/mol
Minimised FF energy 13.23kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.