FAIRMol

OHD_TB2020_32

Pose ID 8788 Compound 968 Pose 209

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.619 kcal/mol/HA) ✓ Good fit quality (FQ -5.91) ✗ Very high strain energy (22.8 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-17.938
kcal/mol
LE
-0.619
kcal/mol/HA
Fit Quality
-5.91
FQ (Leeson)
HAC
29
heavy atoms
MW
434
Da
LogP
4.59
cLogP
Strain ΔE
22.8 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 22.8 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 3 Clashes 10 Severe clashes 1
Final rank6.6762450716022075Score-17.9379
Inter norm-0.722233Intra norm0.0863054
Top1000noExcludedyes
Contacts19H-bonds1
Artifact reasonexcluded; geometry warning; 10 clashes; 1 protein clash; high strain Δ 22.8
ResiduesA:ALA34;A:ARG100;A:ARG59;A:ASP54;A:ILE160;A:ILE47;A:LEU90;A:LEU97;A:MET55;A:NDP301;A:PHE58;A:PHE94;A:PRO91;A:THR184;A:THR86;A:TRP49;A:TYR57;A:VAL32;A:VAL33

Protein summary

223 residues
Protein targetT06Atoms3452
Residues223Chains1
Residue summaryARG:408; VAL:352; LYS:308; LEU:304; PRO:238; ILE:209; GLU:195; THR:182; SER:176; ALA:160; PHE:140; ASN:126; GLY:126; ASP:108; GLN:85; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name8RHTContacts21
PoseOpen native poseH-bonds6
IFP residuesA:ALA34; A:ASP54; A:HIS182; A:ILE160; A:ILE47; A:LEU90; A:LEU97; A:MET55; A:NDP301; A:PHE233; A:PHE58; A:PHE94; A:PRO91; A:SER89; A:THR184; A:THR86; A:TRP49; A:TYR166; A:TYR57; A:VAL32; A:VAL33
Current overlap17Native recall0.81
Jaccard0.74RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
183 2.6524973836816628 -0.93453 -26.7901 0 15 0 0.00 0.00 - no Open
166 3.184967355927311 -0.972893 -27.5669 1 15 0 0.00 0.00 - no Open
182 4.6125044483965 -1.12904 -30.7227 4 17 0 0.00 0.00 - no Open
207 4.723685244314048 -0.759738 -18.573 0 19 17 0.81 0.00 - no Open
98 4.928706460321411 -0.771316 -21.0817 1 12 0 0.00 0.00 - no Open
167 5.865293042808408 -0.980624 -26.822 3 13 0 0.00 0.00 - yes Open
209 6.6762450716022075 -0.722233 -17.9379 1 19 17 0.81 0.00 - yes Current
97 6.758871973745717 -1.00649 -28.4867 1 12 0 0.00 0.00 - yes Open
99 6.9446623186933465 -0.830883 -23.779 1 12 0 0.00 0.00 - yes Open
181 7.556609259784765 -1.16149 -31.6116 3 18 0 0.00 0.00 - yes Open
208 10.990758953446976 -0.742372 -17.8666 0 18 16 0.76 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -17.938kcal/mol
Ligand efficiency (LE) -0.6185kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -5.905
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 29HA

Physicochemical properties

Molecular weight 434.3Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.59
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 22.76kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy -2.38kcal/mol
Minimised FF energy -25.14kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.