FAIRMol

Z266758736

Pose ID 7895 Compound 880 Pose 1308

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-1.656 kcal/mol/HA) ✓ Good fit quality (FQ -14.84) ✗ High strain energy (11.9 kcal/mol) ✗ No H-bonds detected ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-39.734
kcal/mol
LE
-1.656
kcal/mol/HA
Fit Quality
-14.84
FQ (Leeson)
HAC
24
heavy atoms
MW
322
Da
LogP
2.61
cLogP
Strain ΔE
11.9 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 11.9 kcal/mol

Interaction summary

Collapsible panels
H-bonds 0 Hydrophobic 14 π–π 2 Clashes 6 Severe clashes 0
Final rank3.5581947734547623Score-39.7339
Inter norm-0.955682Intra norm-0.699897
Top1000noExcludedno
Contacts15H-bonds0
Artifact reasongeometry warning; 10 clashes; 6 protein contact clashes; very favorable intra outlier; moderate strain Δ 14.3
ResiduesA:ARG17;A:GLY225;A:HIS241;A:LEU188;A:LEU226;A:LEU229;A:MET233;A:NDP302;A:PHE113;A:SER111;A:SER227;A:TYR194;A:VAL230;A:VAL237;D:ARG287

Protein summary

308 residues
Protein targetT04Atoms4210
Residues308Chains3
Residue summaryLEU:494; ALA:421; ARG:384; VAL:368; THR:295; TYR:231; SER:198; PRO:196; ILE:190; LYS:176; ASN:154; GLU:150; GLY:126; PHE:120; HIS:119; ASP:108

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name7PXXContacts19
PoseOpen native poseH-bonds8
IFP residuesA:ARG17; A:ASP181; A:GLY225; A:HIS241; A:LEU188; A:LEU226; A:LEU229; A:LYS198; A:MET233; A:NDP302; A:PHE113; A:PRO115; A:SER111; A:SER112; A:SER227; A:TYR191; A:TYR194; A:VAL230; D:ARG287
Current overlap14Native recall0.74
Jaccard0.70RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

No hydrogen bonds detected for this pose.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1308 3.5581947734547623 -0.955682 -39.7339 0 15 14 0.74 0.00 - no Current
1309 3.8910946977320826 -0.621543 -11.3831 0 12 12 0.63 0.00 - no Open
1304 3.8570512520581826 -0.920966 -17.8731 3 12 12 0.63 0.00 - yes Open
1310 4.340372053343102 -0.887248 -17.065 3 12 12 0.63 0.00 - yes Open
1306 4.926435324388029 -0.960189 -18.1461 2 12 12 0.63 0.00 - yes Open
1303 5.085833785511492 -0.6022 -11.7926 0 11 11 0.58 0.00 - yes Open
1305 8.176416929600043 -0.63778 -5.75832 0 12 12 0.63 0.00 - yes Open
1307 11.393465178559207 -0.729131 -29.3745 1 14 14 0.74 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -39.734kcal/mol
Ligand efficiency (LE) -1.6556kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -14.837
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 24HA

Physicochemical properties

Molecular weight 322.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.61
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 11.91kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 84.20kcal/mol
Minimised FF energy 72.29kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.