FAIRMol

ulfkktlib_3115

Pose ID 6989 Compound 800 Pose 402

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-1.861 kcal/mol/HA) ✓ Good fit quality (FQ -14.56) ✓ Strong H-bond network (16 bonds) ✗ Very high strain energy (22.4 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-31.644
kcal/mol
LE
-1.861
kcal/mol/HA
Fit Quality
-14.56
FQ (Leeson)
HAC
17
heavy atoms
MW
232
Da
LogP
-0.99
cLogP
Strain ΔE
22.4 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 22.4 kcal/mol

Interaction summary

Collapsible panels
H-bonds 16 Hydrophobic 14 π–π 2 Clashes 4 Severe clashes 0
Final rank2.4390965834689524Score-31.6437
Inter norm-1.7656Intra norm-0.0957877
Top1000noExcludedno
Contacts11H-bonds13
Artifact reasongeometry warning; 10 clashes; 4 protein contact clashes; high strain Δ 26.8
ResiduesA:ARG17;A:HIS241;A:LEU188;A:LEU226;A:LEU229;A:LYS198;A:NDP302;A:PHE113;A:SER111;A:TYR194;D:ARG287

Protein summary

308 residues
Protein targetT04Atoms4210
Residues308Chains3
Residue summaryLEU:494; ALA:421; ARG:384; VAL:368; THR:295; TYR:231; SER:198; PRO:196; ILE:190; LYS:176; ASN:154; GLU:150; GLY:126; PHE:120; HIS:119; ASP:108

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: permissive.
Name7PXXContacts19
PoseOpen native poseH-bonds8
IFP residuesA:ARG17; A:ASP181; A:GLY225; A:HIS241; A:LEU188; A:LEU226; A:LEU229; A:LYS198; A:MET233; A:NDP302; A:PHE113; A:PRO115; A:SER111; A:SER112; A:SER227; A:TYR191; A:TYR194; A:VAL230; D:ARG287
Current overlap11Native recall0.58
Jaccard0.58RMSD-
H-bond strict5Strict recall0.83
H-bond same residue+role4Role recall0.80
H-bond same residue4Residue recall0.80

Hydrogen bonds

Mode: permissive. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
937 2.4148800542301965 -1.51727 -25.0218 6 17 0 0.00 0.00 - no Open
402 2.4390965834689524 -1.7656 -31.6437 13 11 11 0.58 0.80 - no Current
589 2.9039670842490644 -1.46649 -27.8436 5 16 0 0.00 0.00 - no Open
1381 3.411492266145569 -1.08304 -18.7427 7 11 0 0.00 0.00 - no Open
588 3.721599539499021 -1.34499 -23.4865 5 17 0 0.00 0.00 - no Open
397 4.289712473650642 -1.50395 -20.6152 13 13 12 0.63 0.80 - no Open
1380 5.544253129452965 -1.16066 -18.8993 7 11 0 0.00 0.00 - no Open
936 4.077173571531417 -1.45164 -24.3531 6 16 0 0.00 0.00 - yes Open
400 4.798722845957986 -1.47873 -24.0411 7 12 12 0.63 0.80 - yes Open
398 5.173685611942922 -1.69808 -28.1451 8 13 13 0.68 0.80 - yes Open
401 6.8246443475113505 -1.38126 -20.7245 9 12 11 0.58 0.40 - yes Open
399 9.27747335375351 -1.38417 -18.3264 10 11 11 0.58 0.80 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -31.644kcal/mol
Ligand efficiency (LE) -1.8614kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -14.556
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 17HA

Physicochemical properties

Molecular weight 232.3Da
Lipinski: ≤ 500 Da
LogP (cLogP) -0.99
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 22.37kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 30.94kcal/mol
Minimised FF energy 8.57kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.