FAIRMol

Z56768366

Pose ID 6151 Compound 274 Pose 2833

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.672 kcal/mol/HA) ✓ Good fit quality (FQ -6.42) ✓ Good H-bonds (4 bonds) ✗ High strain energy (18.7 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-19.493
kcal/mol
LE
-0.672
kcal/mol/HA
Fit Quality
-6.42
FQ (Leeson)
HAC
29
heavy atoms
MW
426
Da
LogP
5.37
cLogP
Strain ΔE
18.7 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 18.7 kcal/mol

Interaction summary

Collapsible panels
H-bonds 4 Hydrophobic 24 π–π 2 Clashes 7 Severe clashes 1
Final rank6.272852567478617Score-19.4932
Inter norm-0.840999Intra norm0.168818
Top1000noExcludedyes
Contacts19H-bonds4
Artifact reasonexcluded; geometry warning; 14 clashes; 1 protein clash; high strain Δ 23.5
ResiduesA:ALA32;A:ARG48;A:ASP52;A:ILE45;A:LEU94;A:MET53;A:NDP301;A:PHE56;A:PRO88;A:SER44;A:SER86;A:THR83;A:TRP47;A:TYR162;A:VAL156;A:VAL30;A:VAL31;A:VAL49;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap15Native recall0.75
Jaccard0.62RMSD-
H-bond strict1Strict recall0.14
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1991 4.819490143075884 -0.90653 -20.8931 5 17 1 0.05 0.00 - no Open
1475 4.962740542105822 -0.773146 -20.2159 1 13 0 0.00 0.00 - no Open
2899 5.299452533493081 -0.876449 -24.5843 1 18 0 0.00 0.00 - no Open
2834 5.542241361549774 -0.914506 -23.3014 2 19 15 0.75 0.20 - no Open
1476 5.561559224811429 -0.838818 -22.236 1 15 0 0.00 0.00 - no Open
1478 5.613641932231067 -0.69062 -16.7448 1 15 0 0.00 0.00 - no Open
1477 5.775010971811956 -0.747567 -19.1127 1 14 0 0.00 0.00 - no Open
2833 6.272852567478617 -0.840999 -19.4932 4 19 15 0.75 0.20 - yes Current
2835 6.338854012321318 -0.96341 -25.2468 1 20 19 0.95 0.20 - yes Open
2832 6.385159074029015 -0.900025 -25.7287 3 16 16 0.80 0.20 - yes Open
2900 7.102127522241116 -0.821543 -23.5752 2 19 0 0.00 0.00 - yes Open
2898 7.495613616474527 -0.846231 -19.0087 6 17 0 0.00 0.00 - yes Open
1992 8.7860722877612 -0.909917 -24.0506 6 16 1 0.05 0.00 - yes Open
1989 9.785917294222623 -0.890102 -20.8213 7 16 1 0.05 0.00 - yes Open
2901 10.45431561116286 -0.82708 -23.7783 2 18 0 0.00 0.00 - yes Open
1990 10.521905467957987 -0.862785 -18.6992 5 17 1 0.05 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -19.493kcal/mol
Ligand efficiency (LE) -0.6722kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.416
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 29HA

Physicochemical properties

Molecular weight 425.9Da
Lipinski: ≤ 500 Da
LogP (cLogP) 5.37
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 18.68kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 71.55kcal/mol
Minimised FF energy 52.87kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.