FAIRMol

Z56768366

Pose ID 2899 Compound 274 Pose 2899

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.848 kcal/mol/HA) ✓ Good fit quality (FQ -8.09) ✗ High strain energy (19.3 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-24.584
kcal/mol
LE
-0.848
kcal/mol/HA
Fit Quality
-8.09
FQ (Leeson)
HAC
29
heavy atoms
MW
426
Da
LogP
5.37
cLogP
Strain ΔE
19.3 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 19.3 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 2 Clashes 7 Severe clashes 0
Final rank5.299452533493081Score-24.5843
Inter norm-0.876449Intra norm0.0287154
Top1000noExcludedno
Contacts18H-bonds1
Artifact reasongeometry warning; 17 clashes; 7 protein contact clashes; high strain Δ 21.6
ResiduesA:ALA10;A:ARG29;A:ASN65;A:GLU31;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:THR137;A:THR57;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap15Native recall0.71
Jaccard0.62RMSD-
H-bond strict1Strict recall0.20
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1991 4.819490143075884 -0.90653 -20.8931 5 17 0 0.00 0.00 - no Open
1475 4.962740542105822 -0.773146 -20.2159 1 13 0 0.00 0.00 - no Open
2899 5.299452533493081 -0.876449 -24.5843 1 18 15 0.71 0.20 - no Current
2834 5.542241361549774 -0.914506 -23.3014 2 19 0 0.00 0.00 - no Open
1476 5.561559224811429 -0.838818 -22.236 1 15 0 0.00 0.00 - no Open
1478 5.613641932231067 -0.69062 -16.7448 1 15 0 0.00 0.00 - no Open
1477 5.775010971811956 -0.747567 -19.1127 1 14 0 0.00 0.00 - no Open
2833 6.272852567478617 -0.840999 -19.4932 4 19 0 0.00 0.00 - yes Open
2835 6.338854012321318 -0.96341 -25.2468 1 20 0 0.00 0.00 - yes Open
2832 6.385159074029015 -0.900025 -25.7287 3 16 0 0.00 0.00 - yes Open
2900 7.102127522241116 -0.821543 -23.5752 2 19 17 0.81 0.00 - yes Open
2898 7.495613616474527 -0.846231 -19.0087 6 17 17 0.81 0.60 - yes Open
1992 8.7860722877612 -0.909917 -24.0506 6 16 0 0.00 0.00 - yes Open
1989 9.785917294222623 -0.890102 -20.8213 7 16 0 0.00 0.00 - yes Open
2901 10.45431561116286 -0.82708 -23.7783 2 18 17 0.81 0.00 - yes Open
1990 10.521905467957987 -0.862785 -18.6992 5 17 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -24.584kcal/mol
Ligand efficiency (LE) -0.8477kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -8.092
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 29HA

Physicochemical properties

Molecular weight 425.9Da
Lipinski: ≤ 500 Da
LogP (cLogP) 5.37
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 19.27kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 73.81kcal/mol
Minimised FF energy 54.54kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.