FAIRMol

Z49638306

Pose ID 5868 Compound 667 Pose 2550

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.764 kcal/mol/HA) ✓ Good fit quality (FQ -7.38) ✓ Strong H-bond network (6 bonds) ✗ High strain energy (11.3 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-22.935
kcal/mol
LE
-0.764
kcal/mol/HA
Fit Quality
-7.38
FQ (Leeson)
HAC
30
heavy atoms
MW
398
Da
LogP
3.86
cLogP
Strain ΔE
11.3 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: mixed
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 11.3 kcal/mol

Interaction summary

Collapsible panels
H-bonds 6 Hydrophobic 24 π–π 2 Clashes 9 Severe clashes 1
Final rank6.798936814767271Score-22.9352
Inter norm-0.774692Intra norm0.0101864
Top1000noExcludedyes
Contacts10H-bonds6
Artifact reasonexcluded; geometry warning; 16 clashes; 1 protein clash; moderate strain Δ 14.0
ResiduesA:ARG97;A:LEU94;A:LYS57;A:LYS90;A:LYS95;A:MET53;A:PHE91;A:PRO88;A:PRO93;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap7Native recall0.35
Jaccard0.30RMSD-
H-bond strict1Strict recall0.14
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1906 4.079634371228655 -0.565681 -19.4954 6 13 0 0.00 0.00 - no Open
1904 4.708431710135203 -0.593572 -18.3879 3 8 0 0.00 0.00 - no Open
2552 5.837738885508001 -0.84258 -26.671 9 11 7 0.35 0.20 - no Open
1374 6.9491310065977725 -1.21986 -37.7354 9 14 0 0.00 0.00 - no Open
1553 7.366388362828268 -0.629821 -20.6491 5 15 0 0.00 0.00 - no Open
1549 8.450095171648368 -0.721285 -24.1068 7 16 0 0.00 0.00 - no Open
1900 6.1831904129384965 -0.71915 -21.2671 8 15 0 0.00 0.00 - yes Open
2548 6.398582763603283 -1.07455 -32.5822 7 12 7 0.35 0.20 - yes Open
2553 6.594207675159006 -0.943559 -27.8785 4 14 12 0.60 0.40 - yes Open
2550 6.798936814767271 -0.774692 -22.9352 6 10 7 0.35 0.20 - yes Current
2549 6.971189554398788 -0.915938 -25.9224 4 14 12 0.60 0.40 - yes Open
1905 7.018537068616989 -0.62468 -21.7228 5 9 0 0.00 0.00 - yes Open
2551 7.033853904040928 -0.845777 -26.335 4 15 13 0.65 0.20 - yes Open
1903 7.414535980267811 -0.629732 -20.3929 5 13 0 0.00 0.00 - yes Open
1901 7.816321035401791 -0.673946 -21.3884 4 13 0 0.00 0.00 - yes Open
1548 8.866106778944213 -0.923782 -27.0501 11 19 0 0.00 0.00 - yes Open
1554 9.058924025034537 -0.757065 -21.7722 11 18 0 0.00 0.00 - yes Open
1902 9.330708255049892 -0.712915 -24.4361 3 13 0 0.00 0.00 - yes Open
1907 9.607718702921597 -0.633204 -22.1142 5 14 0 0.00 0.00 - yes Open
1547 9.80770316554089 -0.668429 -17.3057 5 16 0 0.00 0.00 - yes Open
1552 10.005670834294907 -0.777192 -26.0641 9 19 0 0.00 0.00 - yes Open
1550 10.24519874536975 -1.07037 -31.267 12 18 0 0.00 0.00 - yes Open
1375 10.697110617251491 -1.12097 -37.0518 10 19 0 0.00 0.00 - yes Open
1551 11.621956666465433 -0.756254 -18.4723 7 15 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.935kcal/mol
Ligand efficiency (LE) -0.7645kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.375
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 30HA

Physicochemical properties

Molecular weight 398.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.86
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 11.33kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 109.02kcal/mol
Minimised FF energy 97.69kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.