FAIRMol

OSA_Lib_221

Pose ID 48089 Compound 416 Pose 1124

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.519 kcal/mol/HA) ✓ Good fit quality (FQ -5.32) ✗ Very high strain energy (36.7 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-19.212
kcal/mol
LE
-0.519
kcal/mol/HA
Fit Quality
-5.32
FQ (Leeson)
HAC
37
heavy atoms
MW
504
Da
LogP
1.92
cLogP
Strain ΔE
36.7 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 18 π–π 2 Clashes 5 Severe clashes 0
Final rank5.238380993424386Score-19.2125
Inter norm-0.511812Intra norm-0.0074434
Top1000noExcludedno
Contacts13H-bonds2
Artifact reasongeometry warning; 14 clashes; 5 protein contact clashes; high strain Δ 33.9
ResiduesA:ASN402;A:GLU466;A:GLU467;A:HIS461;A:LEU399;A:PHE396;A:PRO398;A:PRO462;A:SER394;A:SER464;A:SER470;A:THR397;A:THR463

Protein summary

492 residues
Protein targetT20Atoms7539
Residues492Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:264; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name9IFHContacts8
PoseOpen native poseH-bonds2
IFP residuesA:ASN402; A:GLU467; A:LEU399; A:PHE396; A:PRO398; A:SER394; A:SER470; A:THR397
Current overlap8Native recall1.00
Jaccard0.62RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1127 5.038908936669948 -0.365169 -11.4187 1 14 8 1.00 0.00 - no Open
1124 5.238380993424386 -0.511812 -19.2125 2 13 8 1.00 0.00 - no Current
1121 5.5327307586108 -0.350255 -8.02815 1 10 7 0.88 0.00 - no Open
1419 7.356215058806788 -0.552012 -18.9631 2 16 0 0.00 0.00 - no Open
1420 8.047544991033694 -0.724157 -17.5696 2 21 0 0.00 0.00 - no Open
1122 54.57854085204495 -0.438955 -15.2779 3 11 5 0.62 0.00 - no Open
1128 54.58589662623331 -0.313077 -11.3123 1 13 7 0.88 0.00 - no Open
1125 55.18963840714748 -0.394497 -9.98525 1 14 8 1.00 0.00 - no Open
1126 55.480241772929055 -0.397219 -15.0582 2 11 7 0.88 0.00 - no Open
1415 7.484304722717097 -0.64561 -22.563 2 20 0 0.00 0.00 - yes Open
1418 56.574558187707474 -0.539773 -21.1123 2 17 0 0.00 0.00 - yes Open
1123 57.37408623853301 -0.403823 -14.0481 3 13 7 0.88 0.00 - yes Open
1413 57.922520211593174 -0.491911 -16.4026 0 19 0 0.00 0.00 - yes Open
1417 58.78370115098876 -0.513041 -12.5529 1 20 0 0.00 0.00 - yes Open
1416 59.193724545733424 -0.57716 -8.78017 2 17 0 0.00 0.00 - yes Open
1414 59.89441270230394 -0.616844 -19.9818 1 20 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -19.212kcal/mol
Ligand efficiency (LE) -0.5193kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -5.316
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 37HA

Physicochemical properties

Molecular weight 503.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.92
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 36.67kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 168.93kcal/mol
Minimised FF energy 132.26kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.