FAIRMol

OSA_Lib_221

Pose ID 1415 Compound 416 Pose 1415

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.610 kcal/mol/HA) ✓ Good fit quality (FQ -6.24) ✗ Very high strain energy (36.3 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-22.563
kcal/mol
LE
-0.610
kcal/mol/HA
Fit Quality
-6.24
FQ (Leeson)
HAC
37
heavy atoms
MW
504
Da
LogP
1.92
cLogP
Strain ΔE
36.3 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 36.3 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 1 Clashes 7 Severe clashes 1
Final rank7.484304722717097Score-22.563
Inter norm-0.64561Intra norm0.0358
Top1000noExcludedyes
Contacts20H-bonds2
Artifact reasonexcluded; geometry warning; 17 clashes; 1 protein clash; high strain Δ 29.7
ResiduesA:ALA10;A:ASN65;A:ASP22;A:GLN36;A:GLU31;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap18Native recall0.86
Jaccard0.78RMSD-
H-bond strict1Strict recall0.20
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1127 5.038908936669948 -0.365169 -11.4187 1 14 0 0.00 0.00 - no Open
1124 5.238380993424386 -0.511812 -19.2125 2 13 0 0.00 0.00 - no Open
1121 5.5327307586108 -0.350255 -8.02815 1 10 0 0.00 0.00 - no Open
1419 7.356215058806788 -0.552012 -18.9631 2 16 13 0.62 0.20 - no Open
1420 8.047544991033694 -0.724157 -17.5696 2 21 17 0.81 0.00 - no Open
1122 54.57854085204495 -0.438955 -15.2779 3 11 0 0.00 0.00 - no Open
1128 54.58589662623331 -0.313077 -11.3123 1 13 0 0.00 0.00 - no Open
1125 55.18963840714748 -0.394497 -9.98525 1 14 0 0.00 0.00 - no Open
1126 55.480241772929055 -0.397219 -15.0582 2 11 0 0.00 0.00 - no Open
1415 7.484304722717097 -0.64561 -22.563 2 20 18 0.86 0.20 - yes Current
1418 56.574558187707474 -0.539773 -21.1123 2 17 13 0.62 0.20 - yes Open
1123 57.37408623853301 -0.403823 -14.0481 3 13 0 0.00 0.00 - yes Open
1413 57.922520211593174 -0.491911 -16.4026 0 19 16 0.76 0.00 - yes Open
1417 58.78370115098876 -0.513041 -12.5529 1 20 17 0.81 0.20 - yes Open
1416 59.193724545733424 -0.57716 -8.78017 2 17 13 0.62 0.20 - yes Open
1414 59.89441270230394 -0.616844 -19.9818 1 20 17 0.81 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.563kcal/mol
Ligand efficiency (LE) -0.6098kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.243
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 37HA

Physicochemical properties

Molecular weight 503.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.92
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 36.35kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 173.45kcal/mol
Minimised FF energy 137.11kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.