FAIRMol

OHD_TB2020_4

Pose ID 42262 Compound 736 Pose 175

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Acceptable LE (-0.210 kcal/mol/HA) ✓ Good fit quality (FQ -2.29) ✓ Good H-bonds (5 bonds) ✗ Very high strain energy (39.0 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-10.088
kcal/mol
LE
-0.210
kcal/mol/HA
Fit Quality
-2.29
FQ (Leeson)
HAC
48
heavy atoms
MW
665
Da
LogP
3.91
cLogP
Strain ΔE
39.0 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 5 Hydrophobic 24 π–π 3 Clashes 4 Severe clashes 0
Final rank6.275542488399826Score-10.0884
Inter norm-0.230337Intra norm0.0201613
Top1000noExcludedno
Contacts9H-bonds5
Artifact reasongeometry warning; 17 clashes; 4 protein contact clashes; high strain Δ 38.3
ResiduesA:GLU18;A:ILE106;A:LEU17;A:MET113;A:SER109;A:TRP21;A:TYR110;A:VAL53;A:VAL58

Protein summary

493 residues
Protein targetT18Atoms7550
Residues493Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:276; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name6RB5Contacts13
PoseOpen native poseH-bonds0
IFP residuesA:ASP116; A:GLU18; A:GLY112; A:ILE106; A:LEU17; A:MET113; A:SER109; A:THR117; A:THR335; A:TRP21; A:TYR110; A:VAL53; A:VAL58
Current overlap9Native recall0.69
Jaccard0.69RMSD-
H-bond strict0Strict recall-
H-bond same residue+role0Role recall-
H-bond same residue0Residue recall-

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
175 6.275542488399826 -0.230337 -10.0884 5 9 9 0.69 - - no Current
177 6.590816676586569 -0.297682 -14.7996 4 13 10 0.77 - - no Open
122 6.623908820373664 -0.392232 -22.8137 2 16 0 0.00 - - no Open
121 7.38657313809238 -0.321982 -16.1743 3 15 0 0.00 - - no Open
126 7.493058812238245 -0.325898 -13.1866 2 15 0 0.00 - - no Open
174 7.52647633159325 -0.296025 -10.172 1 13 10 0.77 - - no Open
233 7.6319290184965975 -0.406985 -16.0343 1 20 0 0.00 - - no Open
232 8.98296648088481 -0.479979 -19.3352 0 18 0 0.00 - - no Open
130 9.613309366169023 -0.367896 -20.2919 3 13 0 0.00 - - no Open
124 54.90678412804392 -0.446751 -21.3675 4 17 0 0.00 - - no Open
176 55.08095717655768 -0.422474 -17.7921 2 10 10 0.77 - - no Open
179 55.441059436710546 -0.307973 -16.8502 2 9 8 0.62 - - no Open
181 55.4644396591611 -0.309166 -16.1363 1 12 9 0.69 - - no Open
123 56.03713740231415 -0.361384 -18.2614 3 12 0 0.00 - - no Open
129 9.063943532926253 -0.353734 -19.554 3 14 0 0.00 - - yes Open
132 9.21411647823986 -0.319689 -17.7198 2 17 0 0.00 - - yes Open
235 9.632875282411014 -0.40778 -18.0707 0 20 0 0.00 - - yes Open
178 55.54832617343075 -0.355277 -17.897 4 13 11 0.85 - - yes Open
128 55.85736192058398 -0.377757 -22.9116 5 18 0 0.00 - - yes Open
180 56.73329863084768 -0.328082 -16.7695 2 9 8 0.62 - - yes Open
136 57.05145470516479 -0.357664 -15.5151 5 10 0 0.00 - - yes Open
127 57.38136765086828 -0.397318 -18.2109 3 15 0 0.00 - - yes Open
135 57.95106297431023 -0.442919 -19.3927 3 16 0 0.00 - - yes Open
238 58.70619646020666 -0.542864 -22.7362 0 17 0 0.00 - - yes Open
234 58.81723665573986 -0.554031 -24.3529 2 17 0 0.00 - - yes Open
237 59.02381195613867 -0.478612 -20.8327 0 21 0 0.00 - - yes Open
133 59.169384455664925 -0.38743 -14.5111 2 17 0 0.00 - - yes Open
239 59.638485396091426 -0.469957 -20.6378 3 12 0 0.00 - - yes Open
131 59.78931090831168 -0.294202 -15.3285 5 15 0 0.00 - - yes Open
125 61.46460320297299 -0.459124 -21.609 3 17 0 0.00 - - yes Open
236 62.04718782650286 -0.46491 -23.565 2 13 0 0.00 - - yes Open
134 63.28921586966261 -0.401364 -20.4469 2 14 0 0.00 - - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -10.088kcal/mol
Ligand efficiency (LE) -0.2102kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -2.290
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 48HA

Physicochemical properties

Molecular weight 664.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.91
Lipinski: ≤ 5
Rotatable bonds 8

Conformational strain (MMFF94s)

Strain energy (ΔE) 39.05kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 126.67kcal/mol
Minimised FF energy 87.62kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.