FAIRMol

OHD_TB2020_4

Pose ID 3554 Compound 736 Pose 236

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.491 kcal/mol/HA) ✓ Good fit quality (FQ -5.35) ✗ Very high strain energy (63.6 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-23.565
kcal/mol
LE
-0.491
kcal/mol/HA
Fit Quality
-5.35
FQ (Leeson)
HAC
48
heavy atoms
MW
665
Da
LogP
3.91
cLogP
Strain ΔE
63.6 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 63.6 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 2 Clashes 13 Severe clashes 4
Final rank62.04718782650286Score-23.565
Inter norm-0.46491Intra norm-0.0260285
Top1000noExcludedyes
Contacts13H-bonds2
Artifact reasonexcluded; geometry warning; 19 clashes; 4 protein clashes
ResiduesA:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:PHE56;A:PHE91;A:PRO50;A:PRO88;A:THR54;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap11Native recall0.55
Jaccard0.50RMSD-
H-bond strict1Strict recall0.14
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
175 6.275542488399826 -0.230337 -10.0884 5 9 0 0.00 0.00 - no Open
177 6.590816676586569 -0.297682 -14.7996 4 13 0 0.00 0.00 - no Open
122 6.623908820373664 -0.392232 -22.8137 2 16 1 0.05 0.00 - no Open
121 7.38657313809238 -0.321982 -16.1743 3 15 1 0.05 0.00 - no Open
126 7.493058812238245 -0.325898 -13.1866 2 15 0 0.00 0.00 - no Open
174 7.52647633159325 -0.296025 -10.172 1 13 0 0.00 0.00 - no Open
233 7.6319290184965975 -0.406985 -16.0343 1 20 19 0.95 0.00 - no Open
232 8.98296648088481 -0.479979 -19.3352 0 18 14 0.70 0.00 - no Open
130 9.613309366169023 -0.367896 -20.2919 3 13 0 0.00 0.00 - no Open
124 54.90678412804392 -0.446751 -21.3675 4 17 1 0.05 0.00 - no Open
176 55.08095717655768 -0.422474 -17.7921 2 10 0 0.00 0.00 - no Open
179 55.441059436710546 -0.307973 -16.8502 2 9 0 0.00 0.00 - no Open
181 55.4644396591611 -0.309166 -16.1363 1 12 0 0.00 0.00 - no Open
123 56.03713740231415 -0.361384 -18.2614 3 12 1 0.05 0.00 - no Open
129 9.063943532926253 -0.353734 -19.554 3 14 1 0.05 0.00 - yes Open
132 9.21411647823986 -0.319689 -17.7198 2 17 1 0.05 0.00 - yes Open
235 9.632875282411014 -0.40778 -18.0707 0 20 18 0.90 0.00 - yes Open
178 55.54832617343075 -0.355277 -17.897 4 13 0 0.00 0.00 - yes Open
128 55.85736192058398 -0.377757 -22.9116 5 18 0 0.00 0.00 - yes Open
180 56.73329863084768 -0.328082 -16.7695 2 9 0 0.00 0.00 - yes Open
136 57.05145470516479 -0.357664 -15.5151 5 10 1 0.05 0.00 - yes Open
127 57.38136765086828 -0.397318 -18.2109 3 15 1 0.05 0.00 - yes Open
135 57.95106297431023 -0.442919 -19.3927 3 16 1 0.05 0.00 - yes Open
238 58.70619646020666 -0.542864 -22.7362 0 17 15 0.75 0.00 - yes Open
234 58.81723665573986 -0.554031 -24.3529 2 17 15 0.75 0.00 - yes Open
237 59.02381195613867 -0.478612 -20.8327 0 21 17 0.85 0.00 - yes Open
133 59.169384455664925 -0.38743 -14.5111 2 17 1 0.05 0.00 - yes Open
239 59.638485396091426 -0.469957 -20.6378 3 12 10 0.50 0.20 - yes Open
131 59.78931090831168 -0.294202 -15.3285 5 15 0 0.00 0.00 - yes Open
125 61.46460320297299 -0.459124 -21.609 3 17 1 0.05 0.00 - yes Open
236 62.04718782650286 -0.46491 -23.565 2 13 11 0.55 0.20 - yes Current
134 63.28921586966261 -0.401364 -20.4469 2 14 1 0.05 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -23.565kcal/mol
Ligand efficiency (LE) -0.4909kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -5.348
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 48HA

Physicochemical properties

Molecular weight 664.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.91
Lipinski: ≤ 5
Rotatable bonds 8

Conformational strain (MMFF94s)

Strain energy (ΔE) 63.57kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 145.99kcal/mol
Minimised FF energy 82.42kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.