FAIRMol

KB_Leish_36

Pose ID 3836 Compound 109 Pose 518

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-1.028 kcal/mol/HA) ✓ Good fit quality (FQ -9.47) ✓ Strong H-bond network (8 bonds) ✗ Very high strain energy (26.9 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-26.722
kcal/mol
LE
-1.028
kcal/mol/HA
Fit Quality
-9.47
FQ (Leeson)
HAC
26
heavy atoms
MW
349
Da
LogP
2.66
cLogP
Strain ΔE
26.9 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 26.9 kcal/mol

Interaction summary

Collapsible panels
H-bonds 8 Hydrophobic 24 π–π 2 Clashes 5 Severe clashes 0
Final rank4.4601038974391924Score-26.722
Inter norm-0.999455Intra norm-0.0283138
Top1000noExcludedno
Contacts19H-bonds8
Artifact reasongeometry warning; 14 clashes; 5 protein contact clashes; high strain Δ 27.5
ResiduesA:ALA32;A:ARG97;A:ASP52;A:GLY157;A:ILE45;A:LEU94;A:LYS57;A:MET53;A:NDP301;A:PHE55;A:PHE56;A:PHE91;A:THR180;A:TYR162;A:TYR178;A:VAL156;A:VAL30;A:VAL31;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap16Native recall0.80
Jaccard0.70RMSD-
H-bond strict4Strict recall0.57
H-bond same residue+role4Role recall0.80
H-bond same residue4Residue recall0.80

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
486 2.569525141618116 -1.31932 -35.1131 6 16 0 0.00 0.00 - no Open
487 2.5706233481366123 -1.21244 -32.7468 6 16 0 0.00 0.00 - no Open
485 2.6063318911184816 -1.15151 -31.3019 5 16 0 0.00 0.00 - no Open
482 2.746560948394498 -1.24922 -33.3657 4 16 0 0.00 0.00 - no Open
483 3.0881037770074276 -1.16846 -31.7187 4 16 0 0.00 0.00 - no Open
515 3.1059336830861044 -1.03863 -26.8521 8 19 16 0.80 0.80 - no Open
520 3.3538301153175993 -1.08354 -31.3099 4 15 12 0.60 0.20 - no Open
516 3.356499595837022 -1.01808 -26.9593 8 18 13 0.65 0.80 - no Open
484 3.4584880697646083 -1.20344 -32.1171 4 16 0 0.00 0.00 - no Open
471 3.831713010045734 -0.79224 -20.5914 5 13 0 0.00 0.00 - no Open
658 3.9501692319057424 -0.985528 -25.2336 4 15 0 0.00 0.00 - no Open
517 4.064825162545956 -1.07948 -31.1184 6 17 13 0.65 0.80 - no Open
519 4.251722486273004 -1.105 -31.8661 7 17 13 0.65 0.80 - no Open
518 4.4601038974391924 -0.999455 -26.722 8 19 16 0.80 0.80 - no Current
468 4.636093622647474 -0.769462 -22.2181 4 10 0 0.00 0.00 - no Open
625 4.803546563768789 -0.803217 -21.7247 5 12 0 0.00 0.00 - no Open
472 5.396863692971612 -0.903161 -25.3504 6 14 0 0.00 0.00 - no Open
626 5.419036919500527 -0.806911 -21.6887 5 10 0 0.00 0.00 - no Open
578 5.678253723502912 -0.820976 -21.4741 6 18 0 0.00 0.00 - no Open
659 5.111686360577248 -0.945538 -24.3472 3 16 0 0.00 0.00 - yes Open
470 5.9141819054849005 -0.771259 -22.3003 4 10 0 0.00 0.00 - yes Open
467 5.94005831272731 -0.751539 -21.2439 3 10 0 0.00 0.00 - yes Open
579 6.556874896407342 -0.8562 -22.5503 4 19 0 0.00 0.00 - yes Open
624 7.0886128301442595 -0.70565 -21.0809 4 10 0 0.00 0.00 - yes Open
623 7.34512433450863 -0.72924 -20.2579 4 10 0 0.00 0.00 - yes Open
469 8.234825837583921 -0.726875 -18.3807 2 10 0 0.00 0.00 - yes Open
576 8.723183317896952 -0.739238 -19.674 6 12 0 0.00 0.00 - yes Open
577 9.658071359179605 -0.757797 -20.8286 6 15 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -26.722kcal/mol
Ligand efficiency (LE) -1.0278kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -9.469
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 26HA

Physicochemical properties

Molecular weight 349.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.66
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 26.90kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy -112.78kcal/mol
Minimised FF energy -139.68kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.