FAIRMol

KB_Leish_36

Pose ID 28599 Compound 109 Pose 578

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.826 kcal/mol/HA) ✓ Good fit quality (FQ -7.61) ✓ Strong H-bond network (6 bonds) ✗ High strain energy (18.2 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-21.474
kcal/mol
LE
-0.826
kcal/mol/HA
Fit Quality
-7.61
FQ (Leeson)
HAC
26
heavy atoms
MW
350
Da
LogP
2.08
cLogP
Strain ΔE
18.2 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 6 Hydrophobic 9 π–π 0 Clashes 10 Severe clashes 0 ⚠ Hydrophobic exposure 36%
⚠️Partial hydrophobic solvent exposure
37% of hydrophobic surface appears solvent-exposed (7/19 atoms). Partial exposure is common but may limit selectivity and membrane permeability.
Non-polar atoms 19 Buried (contacted) 12 Exposed 7 LogP 2.08 H-bonds 6
Exposed fragments: phenyl (4/6 atoms exposed)phenyl (4/6 atoms exposed)aliphatic chain/group (1 atom exposed)
Final rank5.678253723502912Score-21.4741
Inter norm-0.820976Intra norm-0.00495199
Top1000noExcludedno
Contacts18H-bonds6
Artifact reasongeometry warning; 14 clashes; 10 protein contact clashes; moderate strain Δ 18.7
ResiduesA:ALA283;A:ARG22;A:ARG342;A:ASN20;A:ASP44;A:CYS26;A:GLN341;A:GLU343;A:GLU384;A:LEU25;A:LEU339;A:LEU382;A:PHE284;A:PRO340;A:SER282;A:SER410;A:THR21;A:THR285

Protein summary

398 residues
Protein targetT14Atoms6140
Residues398Chains1
Residue summaryVAL:592; LEU:513; LYS:484; ARG:432; PHE:420; ILE:418; ASP:349; THR:322; TYR:315; PRO:308; GLU:301; ALA:290; SER:253; GLY:217; ASN:210; GLN:170

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name1NJJContacts15
PoseOpen native poseH-bonds7
IFP residuesA:ARG22; A:ARG242; A:ARG337; A:ARG342; A:ASP243; A:ASP385; A:GLN341; A:GLU384; A:LEU25; A:LEU339; A:LEU382; A:PRO340; A:PRO344; A:SER282; A:THR241
Current overlap9Native recall0.60
Jaccard0.38RMSD-
H-bond strict1Strict recall0.17
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

No π–π interactions detected for this pose.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
486 2.569525141618116 -1.31932 -35.1131 6 16 0 0.00 0.00 - no Open
487 2.5706233481366123 -1.21244 -32.7468 6 16 0 0.00 0.00 - no Open
485 2.6063318911184816 -1.15151 -31.3019 5 16 0 0.00 0.00 - no Open
482 2.746560948394498 -1.24922 -33.3657 4 16 0 0.00 0.00 - no Open
483 3.0881037770074276 -1.16846 -31.7187 4 16 0 0.00 0.00 - no Open
515 3.1059336830861044 -1.03863 -26.8521 8 19 0 0.00 0.00 - no Open
520 3.3538301153175993 -1.08354 -31.3099 4 15 0 0.00 0.00 - no Open
516 3.356499595837022 -1.01808 -26.9593 8 18 0 0.00 0.00 - no Open
484 3.4584880697646083 -1.20344 -32.1171 4 16 0 0.00 0.00 - no Open
471 3.831713010045734 -0.79224 -20.5914 5 13 0 0.00 0.00 - no Open
658 3.9501692319057424 -0.985528 -25.2336 4 15 0 0.00 0.00 - no Open
517 4.064825162545956 -1.07948 -31.1184 6 17 0 0.00 0.00 - no Open
519 4.251722486273004 -1.105 -31.8661 7 17 0 0.00 0.00 - no Open
518 4.4601038974391924 -0.999455 -26.722 8 19 0 0.00 0.00 - no Open
468 4.636093622647474 -0.769462 -22.2181 4 10 0 0.00 0.00 - no Open
625 4.803546563768789 -0.803217 -21.7247 5 12 0 0.00 0.00 - no Open
472 5.396863692971612 -0.903161 -25.3504 6 14 0 0.00 0.00 - no Open
626 5.419036919500527 -0.806911 -21.6887 5 10 0 0.00 0.00 - no Open
578 5.678253723502912 -0.820976 -21.4741 6 18 9 0.60 0.20 - no Current
659 5.111686360577248 -0.945538 -24.3472 3 16 0 0.00 0.00 - yes Open
470 5.9141819054849005 -0.771259 -22.3003 4 10 0 0.00 0.00 - yes Open
467 5.94005831272731 -0.751539 -21.2439 3 10 0 0.00 0.00 - yes Open
579 6.556874896407342 -0.8562 -22.5503 4 19 10 0.67 0.20 - yes Open
624 7.0886128301442595 -0.70565 -21.0809 4 10 0 0.00 0.00 - yes Open
623 7.34512433450863 -0.72924 -20.2579 4 10 0 0.00 0.00 - yes Open
469 8.234825837583921 -0.726875 -18.3807 2 10 0 0.00 0.00 - yes Open
576 8.723183317896952 -0.739238 -19.674 6 12 5 0.33 0.20 - yes Open
577 9.658071359179605 -0.757797 -20.8286 6 15 6 0.40 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -21.474kcal/mol
Ligand efficiency (LE) -0.8259kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.610
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 26HA

Physicochemical properties

Molecular weight 350.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.08
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 18.21kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy -124.84kcal/mol
Minimised FF energy -143.05kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.