FAIRMol

KB_HAT_67

Pose ID 3749 Compound 372 Pose 431

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.812 kcal/mol/HA) ✓ Good fit quality (FQ -8.19) ✓ Good H-bonds (3 bonds) ✗ Very high strain energy (53.4 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-28.414
kcal/mol
LE
-0.812
kcal/mol/HA
Fit Quality
-8.19
FQ (Leeson)
HAC
35
heavy atoms
MW
473
Da
LogP
1.61
cLogP
Strain ΔE
53.4 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 53.4 kcal/mol

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 24 π–π 3 Clashes 6 Severe clashes 1
Final rank8.71285521030407Score-28.4143
Inter norm-0.754055Intra norm-0.0577812
Top1000noExcludedyes
Contacts16H-bonds3
Artifact reasonexcluded; geometry warning; 19 clashes; 1 protein clash; high strain Δ 50.8
ResiduesA:ALA32;A:ARG48;A:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:MET53;A:PHE56;A:PHE91;A:PRO50;A:PRO88;A:THR54;A:TRP47;A:VAL49;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap12Native recall0.60
Jaccard0.50RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
362 6.051947950059093 -0.725491 -24.7876 3 19 1 0.05 0.00 - no Open
564 6.435097382084817 -0.76336 -25.367 2 18 0 0.00 0.00 - no Open
562 6.622736186688672 -0.724749 -25.7739 2 20 0 0.00 0.00 - no Open
433 6.929139539328095 -0.831483 -32.4761 2 19 17 0.85 0.40 - no Open
360 7.081412667625094 -0.792379 -30.8426 1 18 1 0.05 0.00 - no Open
432 7.6897862423845496 -0.666396 -18.4122 0 19 18 0.90 0.00 - no Open
563 7.724099824193679 -0.651589 -24.4701 2 15 0 0.00 0.00 - yes Open
434 7.864725185190762 -0.79809 -18.4317 2 20 18 0.90 0.20 - yes Open
431 8.71285521030407 -0.754055 -28.4143 3 16 12 0.60 0.00 - yes Current
565 10.179313852503258 -0.718414 -28.9632 2 19 0 0.00 0.00 - yes Open
430 10.606329162344084 -0.804457 -25.0823 2 16 11 0.55 0.20 - yes Open
361 10.634335700671578 -0.604498 -24.2566 2 12 0 0.00 0.00 - yes Open
363 11.3447361950399 -0.648163 -29.5202 2 12 0 0.00 0.00 - yes Open
435 12.16063322607444 -0.832458 -26.8363 3 15 13 0.65 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -28.414kcal/mol
Ligand efficiency (LE) -0.8118kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -8.189
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 35HA

Physicochemical properties

Molecular weight 472.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.61
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 53.37kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 8.21kcal/mol
Minimised FF energy -45.16kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.