FAIRMol

KB_HAT_67

Pose ID 3748 Compound 372 Pose 430

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.717 kcal/mol/HA) ✓ Good fit quality (FQ -7.23) ✗ Very high strain energy (39.1 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-25.082
kcal/mol
LE
-0.717
kcal/mol/HA
Fit Quality
-7.23
FQ (Leeson)
HAC
35
heavy atoms
MW
473
Da
LogP
1.61
cLogP
Strain ΔE
39.1 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 39.1 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 1 Clashes 12 Severe clashes 2
Final rank10.606329162344084Score-25.0823
Inter norm-0.804457Intra norm0.0878189
Top1000noExcludedyes
Contacts16H-bonds2
Artifact reasonexcluded; geometry warning; 19 clashes; 2 protein clashes; high strain Δ 38.5
ResiduesA:ARG48;A:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:PHE56;A:PHE91;A:PRO88;A:PRO93;A:SER86;A:TRP47;A:VAL49;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap11Native recall0.55
Jaccard0.44RMSD-
H-bond strict2Strict recall0.29
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
362 6.051947950059093 -0.725491 -24.7876 3 19 1 0.05 0.00 - no Open
564 6.435097382084817 -0.76336 -25.367 2 18 0 0.00 0.00 - no Open
562 6.622736186688672 -0.724749 -25.7739 2 20 0 0.00 0.00 - no Open
433 6.929139539328095 -0.831483 -32.4761 2 19 17 0.85 0.40 - no Open
360 7.081412667625094 -0.792379 -30.8426 1 18 1 0.05 0.00 - no Open
432 7.6897862423845496 -0.666396 -18.4122 0 19 18 0.90 0.00 - no Open
563 7.724099824193679 -0.651589 -24.4701 2 15 0 0.00 0.00 - yes Open
434 7.864725185190762 -0.79809 -18.4317 2 20 18 0.90 0.20 - yes Open
431 8.71285521030407 -0.754055 -28.4143 3 16 12 0.60 0.00 - yes Open
565 10.179313852503258 -0.718414 -28.9632 2 19 0 0.00 0.00 - yes Open
430 10.606329162344084 -0.804457 -25.0823 2 16 11 0.55 0.20 - yes Current
361 10.634335700671578 -0.604498 -24.2566 2 12 0 0.00 0.00 - yes Open
363 11.3447361950399 -0.648163 -29.5202 2 12 0 0.00 0.00 - yes Open
435 12.16063322607444 -0.832458 -26.8363 3 15 13 0.65 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -25.082kcal/mol
Ligand efficiency (LE) -0.7166kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.228
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 35HA

Physicochemical properties

Molecular weight 472.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.61
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 39.15kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 5.75kcal/mol
Minimised FF energy -33.40kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.