FAIRMol

OHD_Leishmania_126

Pose ID 3364 Compound 627 Pose 46

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.758 kcal/mol/HA) ✓ Good fit quality (FQ -7.46) ✓ Strong H-bond network (11 bonds) ✗ Very high strain energy (20.7 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-24.270
kcal/mol
LE
-0.758
kcal/mol/HA
Fit Quality
-7.46
FQ (Leeson)
HAC
32
heavy atoms
MW
456
Da
LogP
0.72
cLogP
Strain ΔE
20.7 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 20.7 kcal/mol

Interaction summary

Collapsible panels
H-bonds 11 Hydrophobic 24 π–π 1 Clashes 16 Severe clashes 2
Final rank10.338991350018146Score-24.2699
Inter norm-0.766668Intra norm0.0082325
Top1000noExcludedyes
Contacts22H-bonds11
Artifact reasonexcluded; geometry warning; 16 clashes; 2 protein clashes; high strain Δ 21.9
ResiduesA:ALA32;A:ARG97;A:ASP52;A:ILE45;A:LEU179;A:LEU94;A:LYS57;A:MET53;A:NDP301;A:PHE55;A:PHE56;A:PHE91;A:PRO50;A:PRO88;A:THR180;A:THR54;A:TYR162;A:TYR178;A:VAL156;A:VAL30;A:VAL31;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap18Native recall0.90
Jaccard0.75RMSD-
H-bond strict4Strict recall0.57
H-bond same residue+role3Role recall0.60
H-bond same residue3Residue recall0.60

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
69 3.6077527801455087 -1.00749 -31.9891 6 17 0 0.00 0.00 - no Open
70 3.9202410588473438 -1.13513 -36.4993 8 16 0 0.00 0.00 - no Open
45 5.154007551520005 -0.852745 -25.4636 9 21 18 0.90 0.80 - no Open
46 10.338991350018146 -0.766668 -24.2699 11 22 18 0.90 0.60 - yes Current

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -24.270kcal/mol
Ligand efficiency (LE) -0.7584kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.458
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 32HA

Physicochemical properties

Molecular weight 455.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 0.72
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 20.69kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 43.99kcal/mol
Minimised FF energy 23.30kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.