FAIRMol

Z56958949

Pose ID 3204 Compound 237 Pose 3204

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.779 kcal/mol/HA) ✓ Good fit quality (FQ -7.79) ✗ Very high strain energy (26.6 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-26.483
kcal/mol
LE
-0.779
kcal/mol/HA
Fit Quality
-7.79
FQ (Leeson)
HAC
34
heavy atoms
MW
514
Da
LogP
2.43
cLogP
Strain ΔE
26.6 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 26.6 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 3 Clashes 15 Severe clashes 3
Final rank60.01081702260929Score-26.4833
Inter norm-0.798969Intra norm0.0200472
Top1000noExcludedyes
Contacts19H-bonds1
Artifact reasonexcluded; geometry warning; 11 clashes; 3 protein clashes
ResiduesA:ALA10;A:ASN65;A:ASP22;A:GLN36;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:THR57;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap18Native recall0.86
Jaccard0.82RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
3206 4.948815307706374 -0.684734 -23.3162 1 18 17 0.81 0.00 - no Open
3703 5.418972328285989 -0.620116 -19.2603 3 17 0 0.00 0.00 - no Open
2378 8.222562756337524 -0.79336 -24.4281 7 17 0 0.00 0.00 - no Open
3702 7.61940434743973 -0.745467 -24.4793 4 14 0 0.00 0.00 - yes Open
2376 8.192807940647587 -0.845605 -25.0189 7 18 0 0.00 0.00 - yes Open
2379 10.032734323736642 -0.838117 -20.277 11 16 0 0.00 0.00 - yes Open
3207 10.811693932797503 -0.662537 -18.9743 1 15 11 0.52 0.20 - yes Open
3704 11.093703929308662 -0.700711 -22.7493 4 13 0 0.00 0.00 - yes Open
3205 11.162627935924707 -0.691385 -18.3515 4 19 15 0.71 0.00 - yes Open
3701 59.59594328498775 -0.634484 -20.5254 2 14 0 0.00 0.00 - yes Open
3204 60.01081702260929 -0.798969 -26.4833 1 19 18 0.86 0.00 - yes Current
2377 62.61832617806778 -0.717906 -21.9928 12 17 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -26.483kcal/mol
Ligand efficiency (LE) -0.7789kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.794
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 34HA

Physicochemical properties

Molecular weight 513.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.43
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 26.57kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 29.86kcal/mol
Minimised FF energy 3.30kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.