FAIRMol

Z56900576

Pose ID 2785 Compound 8 Pose 2785

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-1.168 kcal/mol/HA) ✓ Good fit quality (FQ -10.62) ✓ Strong H-bond network (6 bonds) ✗ Very high strain energy (22.8 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-29.206
kcal/mol
LE
-1.168
kcal/mol/HA
Fit Quality
-10.62
FQ (Leeson)
HAC
25
heavy atoms
MW
357
Da
LogP
2.90
cLogP
Strain ΔE
22.8 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 22.8 kcal/mol

Interaction summary

Collapsible panels
H-bonds 6 Hydrophobic 24 π–π 1 Clashes 7 Severe clashes 2
Final rank6.082021025673529Score-29.2064
Inter norm-1.22007Intra norm0.0518152
Top1000noExcludedyes
Contacts18H-bonds5
Artifact reasonexcluded; geometry warning; 4 clashes; 2 protein clashes; high strain Δ 36.4
ResiduesA:ALA10;A:ARG29;A:ASP22;A:GLU31;A:ILE139;A:ILE8;A:LEU23;A:LEU28;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:SER60;A:THR57;A:TRP25;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: permissive.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap13Native recall0.62
Jaccard0.50RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: permissive. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2795 2.2660476124848 -0.849588 -28.2168 2 17 17 0.81 0.20 - no Open
2787 2.7686084214056557 -0.726013 -20.8781 1 18 18 0.86 0.20 - no Open
2791 3.0852186565550435 -0.746411 -21.2571 1 18 18 0.86 0.20 - no Open
2799 3.6423888981391475 -0.715481 -19.2133 1 18 18 0.86 0.20 - no Open
2784 5.664875720951194 -1.07124 -25.6713 5 19 14 0.67 0.20 - no Open
2780 5.845710497953044 -1.13625 -24.527 5 19 14 0.67 0.20 - yes Open
2785 6.082021025673529 -1.22007 -29.2064 5 18 13 0.62 0.20 - yes Current
2794 6.5196138084000985 -0.733943 -19.8468 1 16 15 0.71 0.00 - yes Open
2793 6.604021659825673 -1.08865 -28.4149 5 17 12 0.57 0.20 - yes Open
2783 7.439048407030739 -0.849427 -26.944 5 17 16 0.76 0.20 - yes Open
2797 7.7792432135059455 -1.08679 -28.5021 5 18 14 0.67 0.20 - yes Open
2788 8.07766138806395 -0.989112 -22.0262 6 18 13 0.62 0.20 - yes Open
2789 8.760590011773214 -0.96362 -29.7912 4 19 15 0.71 0.20 - yes Open
2781 9.063335533398318 -1.12244 -24.7856 4 20 15 0.71 0.20 - yes Open
2798 9.331613059388962 -0.746665 -15.0511 8 15 13 0.62 0.20 - yes Open
2792 56.72974551684928 -1.01167 -23.5353 5 19 14 0.67 0.20 - yes Open
2786 58.05530380041594 -0.749477 -18.6166 4 13 8 0.38 0.20 - yes Open
2796 59.321703201143634 -1.03177 -23.363 6 19 14 0.67 0.20 - yes Open
2782 60.07224491906326 -0.968295 -20.6998 5 16 10 0.48 0.20 - yes Open
2790 60.07321101467342 -0.875478 -22.5765 5 19 14 0.67 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -29.206kcal/mol
Ligand efficiency (LE) -1.1683kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -10.621
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 25HA

Physicochemical properties

Molecular weight 357.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.90
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 22.77kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 73.72kcal/mol
Minimised FF energy 50.95kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.