FAIRMol

Z56789391

Pose ID 2517 Compound 89 Pose 2517

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.946 kcal/mol/HA) ✓ Good fit quality (FQ -8.35) ✓ Good H-bonds (3 bonds) ✗ Very high strain energy (42.4 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-21.765
kcal/mol
LE
-0.946
kcal/mol/HA
Fit Quality
-8.35
FQ (Leeson)
HAC
23
heavy atoms
MW
328
Da
LogP
2.88
cLogP
Strain ΔE
42.4 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 42.4 kcal/mol

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 12 π–π 1 Clashes 3 Severe clashes 1
Final rank5.329765757872361Score-21.7654
Inter norm-0.972094Intra norm0.0257714
Top1000noExcludedyes
Contacts15H-bonds3
Artifact reasonexcluded; geometry warning; 8 clashes; 1 protein clash; high strain Δ 43.4
ResiduesA:ALA10;A:ASP22;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:NAP201;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:THR57;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap14Native recall0.67
Jaccard0.64RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2523 3.729762112294257 -0.897843 -18.6811 2 14 14 0.67 0.00 - no Open
2521 4.4503856114985805 -0.839846 -16.6506 2 12 9 0.43 0.00 - no Open
2520 5.335262056321454 -1.14504 -29.5042 3 17 16 0.76 0.40 - no Open
2519 4.2572726577897235 -1.27329 -28.0401 4 14 14 0.67 0.20 - yes Open
2517 5.329765757872361 -0.972094 -21.7654 3 15 14 0.67 0.00 - yes Current
2526 5.375674253869642 -1.03291 -23.9634 2 14 14 0.67 0.00 - yes Open
2525 5.9706404066571475 -1.21239 -24.1089 5 16 16 0.76 0.20 - yes Open
2524 6.992506989180466 -0.95742 -21.7636 1 18 17 0.81 0.20 - yes Open
2518 8.957866303279715 -1.07495 -27.7834 2 16 16 0.76 0.20 - yes Open
2522 10.12363095438683 -0.966963 -21.2769 8 10 6 0.29 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -21.765kcal/mol
Ligand efficiency (LE) -0.9463kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -8.352
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 23HA

Physicochemical properties

Molecular weight 328.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.88
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 42.45kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 79.83kcal/mol
Minimised FF energy 37.38kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.