FAIRMol

OHD_TB2020_48

Pose ID 236 Compound 451 Pose 236

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Good LE (-0.384 kcal/mol/HA) ✓ Good fit quality (FQ -4.11) ✓ Good H-bonds (5 bonds) ✗ Very high strain energy (88.2 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-16.907
kcal/mol
LE
-0.384
kcal/mol/HA
Fit Quality
-4.11
FQ (Leeson)
HAC
44
heavy atoms
MW
611
Da
LogP
-1.02
cLogP
Strain ΔE
88.2 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 88.2 kcal/mol

Interaction summary

Collapsible panels
H-bonds 5 Hydrophobic 24 π–π 0 Clashes 8 Severe clashes 0
Final rank9.659434172653093Score-16.9073
Inter norm-0.476054Intra norm0.0917959
Top1000noExcludedno
Contacts18H-bonds5
Artifact reasongeometry warning; 14 clashes; 8 protein contact clashes; high strain Δ 89.4
ResiduesA:ALA10;A:ASN65;A:ASP22;A:ILE61;A:ILE8;A:LEU23;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO26;A:PRO27;A:PRO62;A:SER60;A:TRP25;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap15Native recall0.71
Jaccard0.62RMSD-
H-bond strict3Strict recall0.60
H-bond same residue+role3Role recall0.60
H-bond same residue3Residue recall0.60

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

No π–π interactions detected for this pose.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
166 7.8000973962403855 -0.405254 -9.34545 4 20 0 0.00 0.00 - no Open
167 8.37163858512793 -0.345489 -14.5393 5 16 0 0.00 0.00 - no Open
236 9.659434172653093 -0.476054 -16.9073 5 18 15 0.71 0.60 - no Current
239 9.586796480250854 -0.544756 -25.3802 7 20 15 0.71 0.80 - yes Open
165 9.922099206829781 -0.57743 -22.1226 7 21 0 0.00 0.00 - yes Open
238 10.408757030452048 -0.500862 -22.7945 3 21 17 0.81 0.40 - yes Open
237 57.32401209749175 -0.578951 -22.2374 9 21 17 0.81 0.80 - yes Open
164 58.48174261162451 -0.401533 -11.3938 9 21 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -16.907kcal/mol
Ligand efficiency (LE) -0.3843kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -4.106
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 44HA

Physicochemical properties

Molecular weight 610.9Da
Lipinski: ≤ 500 Da
LogP (cLogP) -1.02
Lipinski: ≤ 5
Rotatable bonds 10

Conformational strain (MMFF94s)

Strain energy (ΔE) 88.21kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 197.34kcal/mol
Minimised FF energy 109.14kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.