FAIRMol

Z56935963

Pose ID 14428 Compound 1618 Pose 1575

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: queued
Pose metrics recompute is queued in the background.
Metrics cached · SASA missing
T08
Pteridine reductase 1 (PTR1) Trypanosoma brucei
Ligand Z56935963
PDB6RX6

3D complex viewer

Strict H-bonds Permissive H-bonds
Viewer legend
Protein receptor
Pocket residues
Cofactor context
Docked ligand
Overall assessment
Reject No SASA yet
Promising but geometrically suspicious
Binding strong Geometry low Native strong SASA missing
Strain ΔE
42.9 kcal/mol
Protein clashes
7
Internal clashes
2
Native overlap
contact recall 0.79, Jaccard 0.65, H-bond role recall 0.40
Burial
100%
Reason: strain 42.9 kcal/mol
strain ΔE 42.9 kcal/mol 7 protein-contact clashes

Interaction summary

HB 11 HY 24 PI 5 CLASH 2
Final rank4.217Score-30.284
Inter norm-1.329Intra norm0.164
Top1000noExcludedno
Contacts19H-bonds11
Artifact reasongeometry warning; 6 clashes; 7 protein contact clashes; high strain Δ 42.9
Residues
ARG14 ASN175 ASP161 CYS168 LEU208 LEU209 MET163 MET213 NAP301 PHE171 PHE97 PRO167 PRO210 SER207 SER95 TRP221 TYR174 VAL164 VAL206

Protein summary

258 residues
Protein targetT08Atoms3881
Residues258Chains2
Residue summaryLEU:437; VAL:433; ALA:361; ARG:288; ILE:266; GLU:210; LYS:198; SER:198; ASN:182; THR:154; GLN:153; PHE:140; PRO:140; TYR:126; GLY:112; HIS:103

Receptor context

1 kept / 0 excluded
Receptor context filtering: interactions and SASA are computed against protein atoms plus allowed cofactors/ions. Native ligand-like HETATM partners are excluded from scoring.
Kept context 1 Excluded HETATM 0
Kept cofactors / ions
A:NAP301

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
NameTbPTR1_cW_6RX6_ReadyContacts19
PoseOpen native poseHB0
IFP residues
ARG14 ASP161 CYS168 GLY205 LEU208 LEU209 LYS178 MET213 NAP301 PHE171 PHE97 PRO210 PRO99 SER207 SER95 TRP221 TYR174 TYR98 VAL206
Current overlap15Native recall0.79
Jaccard0.65RMSD-
HB strict3Strict recall0.50
HB same residue+role2HB role recall0.40
HB same residue2HB residue recall0.40

HB · H-bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

PI · π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

HY · Hydrophobic contacts

CLASH · Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBCTCT overlapCT recallHB role rec.RMSDExcluded
1580 4.0090486157525005 -1.23767 -31.0171 8 16 15 0.79 0.60 - no Open
1575 4.216856020721941 -1.32914 -30.2835 11 19 15 0.79 0.40 - no Current
1592 4.608546461046636 -0.904944 -16.9271 7 15 14 0.74 0.60 - no Open
1587 4.737810106919343 -1.01697 -20.0824 10 20 15 0.79 0.40 - no Open
1595 4.8654605847064225 -1.31138 -27.2499 12 19 15 0.79 0.60 - no Open
1583 5.615564397178266 -1.09887 -23.7109 11 19 15 0.79 0.40 - no Open
1598 6.167387851197523 -1.00811 -27.0894 8 15 13 0.68 0.60 - no Open
1588 6.266157265092422 -1.04699 -24.7176 7 16 15 0.79 0.60 - no Open
1585 5.374722076766507 -1.08984 -22.8105 4 16 14 0.74 0.20 - yes Open
1581 5.913120864717368 -1.03114 -25.2904 6 18 16 0.84 0.40 - yes Open
1579 6.059584777322205 -1.44502 -29.976 11 18 15 0.79 0.60 - yes Open
1591 6.21589702665084 -0.793403 -21.6499 9 12 9 0.47 0.20 - yes Open
1599 6.96853662992746 -1.2348 -27.4606 12 19 16 0.84 0.60 - yes Open
1594 7.491399332929971 -0.917064 -19.9569 4 10 6 0.32 0.40 - yes Open
1597 7.925203627499189 -1.04999 -29.9225 5 17 14 0.74 0.00 - yes Open
1576 7.930443040877133 -1.28999 -33.4908 8 16 15 0.79 0.60 - yes Open
1601 8.03525322767481 -0.986371 -23.2098 3 17 14 0.74 0.00 - yes Open
1600 8.243357269505164 -1.15919 -29.2886 8 15 14 0.74 0.60 - yes Open
1578 8.36057868967085 -0.997504 -29.6929 5 13 9 0.47 0.60 - yes Open
1590 8.524993999347814 -0.827819 -21.2036 4 11 8 0.42 0.40 - yes Open
1584 9.615994867739026 -1.12669 -20.4656 9 15 13 0.68 0.60 - yes Open
1582 55.213068869816546 -0.935067 -26.7553 7 10 6 0.32 0.60 - yes Open
1596 55.79826082253669 -1.25922 -31.9062 10 17 15 0.79 0.60 - yes Open
1602 56.11746042260958 -0.961668 -27.3851 7 17 14 0.74 0.60 - yes Open
1589 57.965608961708604 -1.03314 -27.723 9 16 16 0.84 0.60 - yes Open
1577 58.42796690225494 -1.18053 -32.9535 11 14 14 0.74 0.60 - yes Open
1593 61.24369911638931 -1.0465 -27.2193 11 14 12 0.63 0.60 - yes Open
1586 65.26605870487273 -0.936415 -14.9554 12 14 13 0.68 0.60 - yes Open

Molecular metrics

RDKit SASA burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
⚠ Not yet computed
Molecular metrics have not been computed for this pose yet. This page now reads only cached values; use a background recompute when you want fresh metrics without slowing the UI.