FAIRMol

Z56815073

Pose ID 12808 Compound 364 Pose 2370

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.880 kcal/mol/HA) ✓ Good fit quality (FQ -8.65) ✗ Very high strain energy (32.8 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-28.148
kcal/mol
LE
-0.880
kcal/mol/HA
Fit Quality
-8.65
FQ (Leeson)
HAC
32
heavy atoms
MW
569
Da
LogP
6.24
cLogP
Strain ΔE
32.8 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 32.8 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 5 Clashes 11 Severe clashes 1
Final rank8.183645678773447Score-28.1484
Inter norm-0.882395Intra norm0.00275864
Top1000noExcludedyes
Contacts15H-bonds2
Artifact reasonexcluded; geometry warning; 13 clashes; 1 protein clash; high strain Δ 31.1
ResiduesA:ARG14;A:CYS168;A:GLU217;A:LEU208;A:LEU209;A:LYS220;A:MET213;A:NAP301;A:PHE171;A:PHE97;A:PRO210;A:SER95;A:TRP221;A:TYR174;A:VAL206

Protein summary

275 residues
Protein targetT07Atoms3932
Residues275Chains3
Residue summaryLEU:437; VAL:433; ALA:361; ARG:288; ILE:266; GLU:210; LYS:198; SER:198; ASN:182; THR:154; GLN:153; PHE:140; PRO:140; TYR:126; GLY:112; HIS:103

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
NameTbPTR1_cW_6RX6_ReadyContacts19
PoseOpen native poseH-bonds6
IFP residuesA:ARG14; A:ASP161; A:CYS168; A:GLY205; A:LEU208; A:LEU209; A:LYS178; A:MET213; A:NAP301; A:PHE171; A:PHE97; A:PRO210; A:PRO99; A:SER207; A:SER95; A:TRP221; A:TYR174; A:TYR98; A:VAL206
Current overlap13Native recall0.68
Jaccard0.62RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2372 4.35739421635852 -0.901914 -30.5487 0 18 14 0.74 0.00 - no Open
1949 5.198949204153766 -0.753505 -21.1708 0 16 0 0.00 0.00 - no Open
3256 6.2634928611964575 -0.933418 -28.8424 4 19 0 0.00 0.00 - no Open
3257 6.455832471385008 -0.821266 -26.9831 1 18 0 0.00 0.00 - no Open
2388 7.774704213900315 -0.802717 -23.7442 1 16 0 0.00 0.00 - no Open
2370 8.183645678773447 -0.882395 -28.1484 2 15 13 0.68 0.00 - yes Current
3255 8.61269293886712 -0.870669 -27.425 0 18 0 0.00 0.00 - yes Open
2387 10.369232843195297 -0.800208 -24.2454 3 18 0 0.00 0.00 - yes Open
2389 12.046434953477675 -0.81696 -27.3427 3 19 0 0.00 0.00 - yes Open
2371 12.536784863271597 -1.04002 -28.6522 3 19 16 0.84 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -28.148kcal/mol
Ligand efficiency (LE) -0.8796kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -8.650
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 32HA

Physicochemical properties

Molecular weight 568.9Da
Lipinski: ≤ 500 Da
LogP (cLogP) 6.24
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 32.80kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 59.38kcal/mol
Minimised FF energy 26.57kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.