FAIRMol

Z104500108

Pose ID 11699 Compound 1327 Pose 1261

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing
T07
Pteridine reductase 1 (PTR1) Trypanosoma brucei
Ligand Z104500108
PDB6RX6

3D complex viewer

Strict H-bonds Permissive H-bonds
Viewer legend
Protein receptor
Pocket residues
Cofactor context
Docked ligand
Overall assessment
Weak No SASA yet
Promising but geometrically suspicious
Binding strong Geometry low Native strong SASA missing
Strain ΔE
15.4 kcal/mol
Protein clashes
0
Internal clashes
12
Native overlap
contact recall 0.74, Jaccard 0.70, H-bond role recall 0.40
Burial
90%
Reason: 12 internal clashes
12 intramolecular clashes
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.785 kcal/mol/HA) ✓ Good fit quality (FQ -7.32) ✓ Strong H-bond network (7 bonds) ✗ Moderate strain (15.4 kcal/mol) ✗ Geometry warnings ✗ Many internal clashes (12) ℹ SASA not computed
Score
-21.193
kcal/mol
LE
-0.785
kcal/mol/HA
Fit Quality
-7.32
FQ (Leeson)
HAC
27
heavy atoms
MW
368
Da
LogP
3.37
cLogP
Strain ΔE
15.4 kcal/mol
SASA buried
computing…

Interaction summary

HB 7 HY 24 PI 4 CLASH 0
Final rank2.353Score-21.193
Inter norm-0.879Intra norm0.094
Top1000noExcludedno
Contacts15H-bonds4
Artifact reasongeometry warning; 12 clashes; 1 protein contact clash; moderate strain Δ 19.8
Residues
ARG14 CYS168 GLY205 LEU208 LEU209 MET163 MET213 NAP301 PHE171 PHE97 PRO210 PRO99 TRP221 TYR174 VAL206

Protein summary

275 residues
Protein targetT07Atoms3932
Residues275Chains3
Residue summaryLEU:437; VAL:433; ALA:361; ARG:288; ILE:266; GLU:210; LYS:198; SER:198; ASN:182; THR:154; GLN:153; PHE:140; PRO:140; TYR:126; GLY:112; HIS:103

Receptor context

1 kept / 0 excluded
Receptor context filtering: interactions and SASA are computed against protein atoms plus allowed cofactors/ions. Native ligand-like HETATM partners are excluded from scoring.
Kept context 1 Excluded HETATM 0
Kept cofactors / ions
A:NAP301

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: permissive.
NameTbPTR1_cW_6RX6_ReadyContacts19
PoseOpen native poseHB0
IFP residues
ARG14 ASP161 CYS168 GLY205 LEU208 LEU209 LYS178 MET213 NAP301 PHE171 PHE97 PRO210 PRO99 SER207 SER95 TRP221 TYR174 TYR98 VAL206
Current overlap14Native recall0.74
Jaccard0.70RMSD-
HB strict3Strict recall0.50
HB same residue+role2HB role recall0.40
HB same residue2HB residue recall0.40

HB · H-bonds

Mode: permissive. Count shows atom-level H-bonds; unique residues in summary: 0.

PI · π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

HY · Hydrophobic contacts

CLASH · Clashes

No clash · clashes detected for this pose.

All stored poses for this docking hit

PoseFinal rankInter normScoreHBCTCT overlapCT recallHB role rec.RMSDExcluded
1261 2.352614741984156 -0.878877 -21.1933 4 15 14 0.74 0.40 - no Current
242 2.447476914358483 -0.908357 -21.8806 4 15 14 0.74 0.40 - no Open
1630 4.715524846739253 -0.640004 -10.8948 2 15 0 0.00 0.00 - no Open
1625 6.074173377966746 -0.80556 -21.7333 9 17 0 0.00 0.00 - no Open
1266 6.824087810079796 -1.00085 -26.9301 6 18 16 0.84 0.60 - no Open
1267 5.514664466722928 -1.05141 -26.1335 6 15 15 0.79 0.40 - yes Open
1264 6.048290580478811 -0.858725 -20.6534 4 17 16 0.84 0.40 - yes Open
1627 6.4706031071443855 -0.772871 -23.0795 9 15 0 0.00 0.00 - yes Open
1263 7.427970208443857 -1.06187 -29.0088 5 20 14 0.74 0.60 - yes Open
1633 8.471081879326855 -0.939358 -18.9139 11 18 0 0.00 0.00 - yes Open
1623 8.8787829524571 -0.557583 -12.8201 9 18 0 0.00 0.00 - yes Open
1632 9.29755773218558 -0.659444 -17.2243 9 16 0 0.00 0.00 - yes Open
1622 11.622027407212617 -0.807135 -21.8272 9 15 0 0.00 0.00 - yes Open
1619 12.158462089191984 -0.59039 -11.4685 9 15 0 0.00 0.00 - yes Open
1620 12.483486148698473 -0.809041 -11.3455 8 14 0 0.00 0.00 - yes Open
1628 57.20569199706915 -0.766764 -11.9344 7 15 0 0.00 0.00 - yes Open
1626 57.29859762330209 -0.682621 -10.3988 11 17 0 0.00 0.00 - yes Open
1262 58.043689460527446 -0.991328 -20.1182 5 15 12 0.63 0.40 - yes Open
1629 59.530653812090854 -0.715619 -16.0066 7 16 0 0.00 0.00 - yes Open
1631 59.74134408162453 -0.617577 -14.5273 8 17 0 0.00 0.00 - yes Open
1621 60.97370136158834 -0.801387 -20.8088 11 16 0 0.00 0.00 - yes Open
1624 61.275380495880434 -0.764099 -18.1143 10 16 0 0.00 0.00 - yes Open
1265 62.718700127462505 -1.0153 -21.1272 7 20 15 0.79 0.20 - yes Open

Molecular metrics

RDKit SASA burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -21.193kcal/mol
Ligand efficiency (LE) -0.7849kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.323
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 27HA

Physicochemical properties

Molecular weight 368.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.37
Lipinski: ≤ 5
Rotatable bonds 8

Conformational strain (MMFF94s)

Strain energy (ΔE) 15.36kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 61.05kcal/mol
Minimised FF energy 45.70kcal/mol

SASA & burial

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate SASA burial metrics without blocking the page.