FAIRMol

NMT-TY0959

Pose ID 11302 Compound 550 Pose 864

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing
T07
Pteridine reductase 1 (PTR1) Trypanosoma brucei
Ligand NMT-TY0959
PDB6RX6

3D complex viewer

Strict H-bonds Permissive H-bonds
Viewer legend
Protein receptor
Pocket residues
Cofactor context
Docked ligand
Overall assessment
Weak No SASA yet
Weak or marginal quality
Binding strong Geometry medium Native strong SASA missing
Strain ΔE
31.4 kcal/mol
Protein clashes
3
Internal clashes
4
Native overlap
contact recall 0.68, Jaccard 0.65, H-bond role recall 0.60
Burial
100%
Reason: no major geometry red flags detected
3 protein-contact clashes 4 intramolecular clashes
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-1.047 kcal/mol/HA) ✓ Good fit quality (FQ -9.77) ✓ Strong H-bond network (6 bonds) ✗ Very high strain energy (31.4 kcal/mol) ✗ Geometry warnings ✗ Many internal clashes (11) ✗ Excluded by docking heuristics ℹ SASA not computed
Score
-28.263
kcal/mol
LE
-1.047
kcal/mol/HA
Fit Quality
-9.77
FQ (Leeson)
HAC
27
heavy atoms
MW
403
Da
LogP
2.27
cLogP
Strain ΔE
31.4 kcal/mol
SASA buried
computing…

Interaction summary

HB 6 HY 24 PI 4 CLASH 4
Final rank11.449Score-28.263
Inter norm-1.058Intra norm0.011
Top1000noExcludedyes
Contacts14H-bonds6
Artifact reasonexcluded; geometry warning; 11 clashes; 3 protein clashes; high strain Δ 36.4
Residues
ARG14 CYS168 LEU208 LEU209 MET169 MET213 NAP301 PHE171 PHE97 PRO210 SER207 SER95 TRP221 TYR174

Protein summary

275 residues
Protein targetT07Atoms3932
Residues275Chains3
Residue summaryLEU:437; VAL:433; ALA:361; ARG:288; ILE:266; GLU:210; LYS:198; SER:198; ASN:182; THR:154; GLN:153; PHE:140; PRO:140; TYR:126; GLY:112; HIS:103

Receptor context

1 kept / 0 excluded
Receptor context filtering: interactions and SASA are computed against protein atoms plus allowed cofactors/ions. Native ligand-like HETATM partners are excluded from scoring.
Kept context 1 Excluded HETATM 0
Kept cofactors / ions
A:NAP301

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
NameTbPTR1_cW_6RX6_ReadyContacts19
PoseOpen native poseHB0
IFP residues
ARG14 ASP161 CYS168 GLY205 LEU208 LEU209 LYS178 MET213 NAP301 PHE171 PHE97 PRO210 PRO99 SER207 SER95 TRP221 TYR174 TYR98 VAL206
Current overlap13Native recall0.68
Jaccard0.65RMSD-
HB strict4Strict recall0.67
HB same residue+role3HB role recall0.60
HB same residue3HB residue recall0.60

HB · H-bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

PI · π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

HY · Hydrophobic contacts

CLASH · Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBCTCT overlapCT recallHB role rec.RMSDExcluded
976 3.725963286202594 -1.30957 -33.6603 12 15 14 0.74 0.40 - no Open
2327 4.096964183561333 -1.05228 -30.182 4 18 0 0.00 0.00 - no Open
3072 4.4521658121106125 -0.766941 -20.0969 5 16 0 0.00 0.00 - no Open
744 4.523667717252291 -1.25191 -32.6226 7 21 0 0.00 0.00 - no Open
2968 4.5596903350546825 -1.0015 -27.2048 10 16 0 0.00 0.00 - no Open
784 4.630887405506052 -0.901881 -22.2926 2 13 0 0.00 0.00 - no Open
3070 4.832518365754668 -0.893622 -24.2732 6 18 0 0.00 0.00 - no Open
1245 4.890463367622139 -1.00246 -29.0104 9 15 0 0.00 0.00 - no Open
1539 4.911094108151013 -0.728068 -18.0762 6 9 0 0.00 0.00 - no Open
789 5.131472184269517 -0.926251 -24.8853 2 13 0 0.00 0.00 - no Open
787 5.548281609924738 -0.852751 -21.3044 1 12 0 0.00 0.00 - no Open
2966 5.7005705101682045 -0.889641 -22.6382 7 15 0 0.00 0.00 - no Open
1196 5.899769271662714 -0.962721 -26.2813 4 18 0 0.00 0.00 - no Open
1542 6.3127925535131055 -0.843132 -22.6989 8 16 0 0.00 0.00 - no Open
861 6.377997963385409 -0.94121 -26.6787 3 15 14 0.74 0.20 - no Open
980 6.551701347950366 -1.1173 -25.4413 9 15 13 0.68 0.40 - no Open
786 6.808597452705019 -0.914363 -21.2318 2 13 0 0.00 0.00 - no Open
2964 6.886427946353083 -0.856264 -23.0552 5 17 0 0.00 0.00 - no Open
1010 7.408671293611844 -1.12176 -28.2281 10 20 0 0.00 0.00 - no Open
992 7.41031777306122 -0.9552 -20.4555 4 16 0 0.00 0.00 - no Open
3069 5.08222974628391 -0.901066 -24.1454 6 15 0 0.00 0.00 - yes Open
1199 5.3054315442508475 -0.875079 -22.9236 3 20 0 0.00 0.00 - yes Open
788 5.595288997168039 -0.880209 -24.3479 2 13 0 0.00 0.00 - yes Open
2963 5.664947554071436 -1.02855 -27.026 8 17 0 0.00 0.00 - yes Open
1541 5.975886762699564 -0.76536 -19.0371 6 13 0 0.00 0.00 - yes Open
1011 6.101892322098901 -1.08066 -26.4646 8 16 0 0.00 0.00 - yes Open
1198 6.292092672987181 -0.930634 -26.173 10 14 0 0.00 0.00 - yes Open
2323 6.313896537521306 -0.894306 -22.1695 2 15 0 0.00 0.00 - yes Open
2326 6.514535612975343 -0.987141 -21.3955 4 17 0 0.00 0.00 - yes Open
743 6.7538176312691025 -1.19073 -29.8295 8 20 0 0.00 0.00 - yes Open
1538 6.857035124312529 -0.776205 -17.5182 6 14 0 0.00 0.00 - yes Open
1194 7.113236760855778 -0.866426 -22.0336 3 15 0 0.00 0.00 - yes Open
2965 7.552429621926622 -0.914149 -25.3534 9 16 0 0.00 0.00 - yes Open
1537 7.650336675401466 -0.796181 -20.743 6 14 0 0.00 0.00 - yes Open
1543 7.652962705554535 -0.850128 -21.98 8 14 0 0.00 0.00 - yes Open
1009 7.827333489442097 -1.0222 -26.8251 7 24 0 0.00 0.00 - yes Open
785 7.992331552127431 -0.805383 -20.8258 3 13 0 0.00 0.00 - yes Open
1195 8.088001666503295 -0.949734 -24.1142 8 15 0 0.00 0.00 - yes Open
745 8.088052672982203 -1.21569 -31.7738 9 20 0 0.00 0.00 - yes Open
978 8.239652498200421 -1.22448 -31.8995 9 15 11 0.58 0.60 - yes Open
3073 8.245653336522212 -0.924839 -25.7132 8 13 0 0.00 0.00 - yes Open
979 8.31593892914662 -1.21839 -28.3093 10 17 13 0.68 0.40 - yes Open
1013 8.470703369671075 -1.0732 -28.8909 14 20 0 0.00 0.00 - yes Open
1244 8.490601006534428 -0.960305 -25.4464 8 18 0 0.00 0.00 - yes Open
1193 8.505495413417659 -0.902642 -22.8728 8 15 0 0.00 0.00 - yes Open
1197 8.642741608851852 -1.08116 -27.9486 7 17 0 0.00 0.00 - yes Open
1008 8.76423981282301 -0.935135 -25.7853 9 21 0 0.00 0.00 - yes Open
2325 8.796722728576952 -1.07172 -28.3571 5 20 0 0.00 0.00 - yes Open
1540 8.925783600326923 -0.742464 -15.947 8 15 0 0.00 0.00 - yes Open
746 8.968390532111323 -1.17375 -31.7016 10 20 0 0.00 0.00 - yes Open
3071 8.99057834845964 -0.784302 -15.8048 5 12 0 0.00 0.00 - yes Open
2967 9.170157968850281 -0.976077 -27.002 9 18 0 0.00 0.00 - yes Open
2328 9.278822190931775 -0.959989 -25.8197 7 10 0 0.00 0.00 - yes Open
862 9.295844880558743 -1.14475 -30.9484 7 15 14 0.74 0.40 - yes Open
993 9.45080372061048 -0.770327 -18.0331 3 17 0 0.00 0.00 - yes Open
977 9.585854727229679 -1.22911 -31.2395 6 17 12 0.63 0.20 - yes Open
1246 9.610255930126277 -1.00961 -29.4309 9 12 0 0.00 0.00 - yes Open
3068 10.121919958869 -0.80158 -21.1804 8 16 0 0.00 0.00 - yes Open
1012 10.16499353802062 -1.1408 -30.4082 8 22 0 0.00 0.00 - yes Open
3074 10.225125480925996 -0.816289 -20.1152 8 14 0 0.00 0.00 - yes Open
863 10.588319598395609 -1.01589 -29.1184 6 16 14 0.74 0.60 - yes Open
747 10.644785406466566 -1.0815 -28.7503 8 21 0 0.00 0.00 - yes Open
2324 10.987677217752333 -0.897714 -26.3186 6 17 0 0.00 0.00 - yes Open
991 11.328862090659927 -0.958753 -24.3683 6 21 0 0.00 0.00 - yes Open
990 11.388062374646408 -0.983958 -24.6706 6 21 0 0.00 0.00 - yes Open
864 11.448545983706115 -1.05756 -28.2634 6 14 13 0.68 0.60 - yes Current
749 12.003813205196298 -1.04534 -29.1571 11 21 0 0.00 0.00 - yes Open
748 13.299026769487188 -1.26034 -34.3636 9 22 0 0.00 0.00 - yes Open

Molecular metrics

RDKit SASA burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -28.263kcal/mol
Ligand efficiency (LE) -1.0468kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -9.766
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 27HA

Physicochemical properties

Molecular weight 403.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.27
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 31.39kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 17.58kcal/mol
Minimised FF energy -13.82kcal/mol

SASA & burial

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate SASA burial metrics without blocking the page.