FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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3 compounds in matrix 6 best compound-target hits listed 6 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T09T15T16T17T20
Z56958949
[H]N(C(=O)CN1C(=O)/C(=C2/SC(=S)N([C@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccccc1
0.883 0.840 3 0.88 0.86 0.78
Z56958949
[H]N(C(=O)CN1C(=O)/C(=C2\SC(=S)N([C@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccccc1
0.855 0.820 2 0.85 0.78
Z56958949
[H]N(C(=O)CN1C(=O)/C(=C2\SC(=S)N([C@@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccccc1
0.786 0.786 1 0.79

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z56958949
[H]N(C(=O)CN1C(=O)/C(=C2/SC(=S)N([C@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccccc1
T09
native IFP available
T09
selection_import_t09
0.883 1.000 0.667 native_similarity final_rank_score -29.412 -0.893982 17 3 Pose
Z56958949
[H]N(C(=O)CN1C(=O)/C(=C2/SC(=S)N([C@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccccc1
T15
native IFP available
T15
selection_import_t15
0.859 1.000 0.597 native_similarity final_rank_score -24.4793 -0.745467 14 4 Pose
Z56958949
[H]N(C(=O)CN1C(=O)/C(=C2\SC(=S)N([C@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccccc1
T02
native IFP available
T02
selection_import_t02
0.855 1.000 0.584 native_similarity final_rank_score -26.4833 -0.798969 19 1 Pose
Z56958949
[H]N(C(=O)CN1C(=O)/C(=C2\SC(=S)N([C@@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccccc1
T17
native IFP available
T17
selection_import_t17
0.786 1.000 0.389 native_similarity final_rank_score -24.8825 -0.727728 19 4 Pose
Z56958949
[H]N(C(=O)CN1C(=O)/C(=C2\SC(=S)N([C@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccccc1
T20
native IFP available
T20
selection_import_t20
0.785 1.000 0.385 native_similarity final_rank_score -20.3366 -0.618611 13 3 Pose
Z56958949
[H]N(C(=O)CN1C(=O)/C(=C2/SC(=S)N([C@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccccc1
T16
native IFP available
T16
selection_import_t16
0.779 1.000 0.368 native_similarity final_rank_score -23.5172 -0.689074 15 1 Pose