FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 6 best compound-target hits listed 6 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T03T07T09T11T19
Z54938583
[H]N([H])n1c(S[C@H](C(=O)c2cn([H])c3ccccc23)c2ccccc2)nnc1-c1ccc(OC)c(OC)c1
0.853 0.823 4 0.85 0.79 0.81 0.84
Z54938583
[H]N([H])n1c(S[C@@H](C(=O)c2cn([H])c3ccccc23)c2ccccc2)nnc1-c1ccc(OC)c(OC)c1
0.851 0.801 2 0.85 0.75

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z54938583
[H]N([H])n1c(S[C@H](C(=O)c2cn([H])c3ccccc23)c2ccccc2)nnc1-c1ccc(OC)c(OC)c1
T01
native IFP available
T01
selection_import_t01
0.853 1.000 0.579 native_similarity final_rank_score -23.2003 -0.762299 17 4 Pose
Z54938583
[H]N([H])n1c(S[C@@H](C(=O)c2cn([H])c3ccccc23)c2ccccc2)nnc1-c1ccc(OC)c(OC)c1
T07
native IFP available
T07
selection_import_t07
0.851 1.000 0.574 native_similarity final_rank_score -31.2638 -0.859212 19 8 Pose
Z54938583
[H]N([H])n1c(S[C@H](C(=O)c2cn([H])c3ccccc23)c2ccccc2)nnc1-c1ccc(OC)c(OC)c1
T11
native IFP available
T11
selection_import_t11
0.844 1.000 0.555 native_similarity final_rank_score -23.4943 -0.691369 14 4 Pose
Z54938583
[H]N([H])n1c(S[C@H](C(=O)c2cn([H])c3ccccc23)c2ccccc2)nnc1-c1ccc(OC)c(OC)c1
T09
native IFP available
T09
selection_import_t09
0.805 1.000 0.444 native_similarity final_rank_score -19.8565 -0.735224 17 6 Pose
Z54938583
[H]N([H])n1c(S[C@H](C(=O)c2cn([H])c3ccccc23)c2ccccc2)nnc1-c1ccc(OC)c(OC)c1
T03
native IFP available
T03
selection_import_t03
0.791 1.000 0.403 native_similarity final_rank_score -25.0279 -0.814168 18 3 Pose
Z54938583
[H]N([H])n1c(S[C@@H](C(=O)c2cn([H])c3ccccc23)c2ccccc2)nnc1-c1ccc(OC)c(OC)c1
T19
native IFP available
T19
selection_import_t19
0.752 1.000 0.291 native_similarity final_rank_score -32.066 -0.992974 24 9 Pose