FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 13 best compound-target hits listed 13 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T03T05T07T09T10T11T12T14T17T20T21T22
Z49604116
[H]Oc1ccc(/C=N\N([H])C(=O)c2cccc(S(=O)(=O)N(CC)CC)c2)c(O[H])c1O[H]
0.940 0.852 10 0.85 0.78 0.80 0.89 0.81 0.89 0.80 0.91 0.94 0.84
Z49604116
[H]Oc1ccc(/C=N/N=C(\O)c2cccc(S(=O)(=O)N(CC)CC)c2)c(O[H])c1O[H]
0.934 0.893 3 0.93 0.85 0.90

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z49604116
[H]Oc1ccc(/C=N\N([H])C(=O)c2cccc(S(=O)(=O)N(CC)CC)c2)c(O[H])c1O[H]
T21
native IFP available
T21
selection_import_t21
0.940 1.000 0.828 native_similarity final_rank_score -30.4779 -0.995794 16 16 Pose
Z49604116
[H]Oc1ccc(/C=N/N=C(\O)c2cccc(S(=O)(=O)N(CC)CC)c2)c(O[H])c1O[H]
T10
native IFP available
T10
selection_import_t10
0.934 1.000 0.812 native_similarity final_rank_score -25.8494 -0.982614 19 11 Pose
Z49604116
[H]Oc1ccc(/C=N\N([H])C(=O)c2cccc(S(=O)(=O)N(CC)CC)c2)c(O[H])c1O[H]
T17
native IFP available
T17
selection_import_t17
0.908 1.000 0.737 native_similarity final_rank_score -19.0924 -0.799965 14 7 Pose
Z49604116
[H]Oc1ccc(/C=N/N=C(\O)c2cccc(S(=O)(=O)N(CC)CC)c2)c(O[H])c1O[H]
T20
native IFP available
T20
selection_import_t20
0.898 1.000 0.710 native_similarity final_rank_score -18.59 -0.736984 11 11 Pose
Z49604116
[H]Oc1ccc(/C=N\N([H])C(=O)c2cccc(S(=O)(=O)N(CC)CC)c2)c(O[H])c1O[H]
T07
native IFP available
T07
selection_import_t07
0.891 1.000 0.690 native_similarity final_rank_score -37.0671 -1.25157 18 11 Pose
Z49604116
[H]Oc1ccc(/C=N\N([H])C(=O)c2cccc(S(=O)(=O)N(CC)CC)c2)c(O[H])c1O[H]
T12
native IFP available
T12
selection_import_t12
0.891 1.000 0.687 native_similarity final_rank_score -20.8301 -0.967244 17 10 Pose
Z49604116
[H]Oc1ccc(/C=N\N([H])C(=O)c2cccc(S(=O)(=O)N(CC)CC)c2)c(O[H])c1O[H]
T02
native IFP available
T02
selection_import_t02
0.855 1.000 0.584 native_similarity final_rank_score -19.4906 -0.946596 19 5 Pose
Z49604116
[H]Oc1ccc(/C=N/N=C(\O)c2cccc(S(=O)(=O)N(CC)CC)c2)c(O[H])c1O[H]
T11
native IFP available
T11
selection_import_t11
0.846 1.000 0.559 native_similarity final_rank_score -28.6177 -0.895643 10 9 Pose
Z49604116
[H]Oc1ccc(/C=N\N([H])C(=O)c2cccc(S(=O)(=O)N(CC)CC)c2)c(O[H])c1O[H]
T22
native IFP available
T22
selection_import_t22
0.843 1.000 0.550 native_similarity final_rank_score -25.6203 -1.14157 23 16 Pose
Z49604116
[H]Oc1ccc(/C=N\N([H])C(=O)c2cccc(S(=O)(=O)N(CC)CC)c2)c(O[H])c1O[H]
T09
native IFP available
T09
selection_import_t09
0.813 1.000 0.465 native_similarity final_rank_score -24.6787 -0.928563 19 6 Pose
Z49604116
[H]Oc1ccc(/C=N\N([H])C(=O)c2cccc(S(=O)(=O)N(CC)CC)c2)c(O[H])c1O[H]
T05
native IFP available
T05
selection_import_t05
0.803 1.000 0.436 native_similarity final_rank_score -32.5527 -1.00866 10 9 Pose
Z49604116
[H]Oc1ccc(/C=N\N([H])C(=O)c2cccc(S(=O)(=O)N(CC)CC)c2)c(O[H])c1O[H]
T14
native IFP available
T14
selection_import_t14
0.797 1.000 0.420 native_similarity final_rank_score -26.6114 -0.9842 14 9 Pose
Z49604116
[H]Oc1ccc(/C=N\N([H])C(=O)c2cccc(S(=O)(=O)N(CC)CC)c2)c(O[H])c1O[H]
T03
native IFP available
T03
selection_import_t03
0.782 1.000 0.377 native_similarity final_rank_score -32.7967 -1.10461 14 11 Pose