FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 13 best compound-target hits listed 13 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T06T07T09T10T11T12T14T17T18T19T21T22
Z18509545
[H]N(Cc1ccc2c(c1)OCO2)C(=O)[C@H](C)N1c2cccc3cccc(c23)S1(=O)=O
0.954 0.861 7 0.86 0.82 0.83 0.89 0.88 0.95 0.79
Z18509545
[H]N(Cc1ccc2c(c1)OCO2)C(=O)[C@@H](C)N1c2cccc3cccc(c23)S1(=O)=O
0.934 0.810 6 0.79 0.76 0.87 0.78 0.73 0.93

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z18509545
[H]N(Cc1ccc2c(c1)OCO2)C(=O)[C@H](C)N1c2cccc3cccc(c23)S1(=O)=O
T12
native IFP available
T12
selection_import_t12
0.954 1.000 0.870 native_similarity final_rank_score -26.9312 -1.03918 16 11 Pose
Z18509545
[H]N(Cc1ccc2c(c1)OCO2)C(=O)[C@@H](C)N1c2cccc3cccc(c23)S1(=O)=O
T21
native IFP available
T21
selection_import_t21
0.934 1.000 0.812 native_similarity final_rank_score -23.3667 -0.865048 15 12 Pose
Z18509545
[H]N(Cc1ccc2c(c1)OCO2)C(=O)[C@H](C)N1c2cccc3cccc(c23)S1(=O)=O
T10
native IFP available
T10
selection_import_t10
0.889 1.000 0.682 native_similarity final_rank_score -25.6601 -0.930167 14 13 Pose
Z18509545
[H]N(Cc1ccc2c(c1)OCO2)C(=O)[C@H](C)N1c2cccc3cccc(c23)S1(=O)=O
T11
native IFP available
T11
selection_import_t11
0.881 1.000 0.661 native_similarity final_rank_score -23.2766 -0.820794 13 6 Pose
Z18509545
[H]N(Cc1ccc2c(c1)OCO2)C(=O)[C@@H](C)N1c2cccc3cccc(c23)S1(=O)=O
T17
native IFP available
T17
selection_import_t17
0.868 1.000 0.622 native_similarity final_rank_score -21.3765 -0.7654 14 3 Pose
Z18509545
[H]N(Cc1ccc2c(c1)OCO2)C(=O)[C@H](C)N1c2cccc3cccc(c23)S1(=O)=O
T02
native IFP available
T02
selection_import_t02
0.860 1.000 0.600 native_similarity final_rank_score -25.8221 -0.957756 18 1 Pose
Z18509545
[H]N(Cc1ccc2c(c1)OCO2)C(=O)[C@H](C)N1c2cccc3cccc(c23)S1(=O)=O
T09
native IFP available
T09
selection_import_t09
0.832 1.000 0.519 native_similarity final_rank_score -21.9547 -0.871795 17 2 Pose
Z18509545
[H]N(Cc1ccc2c(c1)OCO2)C(=O)[C@H](C)N1c2cccc3cccc(c23)S1(=O)=O
T07
native IFP available
T07
selection_import_t07
0.823 1.000 0.496 native_similarity final_rank_score -31.388 -1.10204 17 3 Pose
Z18509545
[H]N(Cc1ccc2c(c1)OCO2)C(=O)[C@@H](C)N1c2cccc3cccc(c23)S1(=O)=O
T06
native IFP available
T06
selection_import_t06
0.791 1.000 0.402 native_similarity final_rank_score -23.3199 -0.904267 16 0 Pose
Z18509545
[H]N(Cc1ccc2c(c1)OCO2)C(=O)[C@H](C)N1c2cccc3cccc(c23)S1(=O)=O
T22
native IFP available
T22
selection_import_t22
0.785 1.000 0.386 native_similarity final_rank_score -28.9651 -1.08923 21 7 Pose
Z18509545
[H]N(Cc1ccc2c(c1)OCO2)C(=O)[C@@H](C)N1c2cccc3cccc(c23)S1(=O)=O
T18
native IFP available
T18
selection_import_t18
0.777 1.000 0.362 native_similarity final_rank_score -19.7334 -0.711603 13 6 Pose
Z18509545
[H]N(Cc1ccc2c(c1)OCO2)C(=O)[C@@H](C)N1c2cccc3cccc(c23)S1(=O)=O
T14
native IFP available
T14
selection_import_t14
0.765 1.000 0.327 native_similarity final_rank_score -21.3729 -0.786036 14 4 Pose
Z18509545
[H]N(Cc1ccc2c(c1)OCO2)C(=O)[C@@H](C)N1c2cccc3cccc(c23)S1(=O)=O
T19
native IFP available
T19
selection_import_t19
0.725 1.000 0.215 native_similarity final_rank_score -32.3995 -1.0974 19 6 Pose