FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 7 best compound-target hits listed 7 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T03T09T15T18T20
Z1820095916
[H]N(Cc1cccs1)C(=O)C1CCN(c2n(Cc3cc(C)ccc3C)c3ccccc3[n+]2[H])CC1
0.864 0.814 6 0.84 0.86 0.79 0.82 0.79 0.76
Z1820095916
[H]N(Cc1cccs1)C(=O)C1CCN(c2nc3ccccc3n2Cc2cc(C)ccc2C)CC1
0.812 0.812 1 0.81

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z1820095916
[H]N(Cc1cccs1)C(=O)C1CCN(c2n(Cc3cc(C)ccc3C)c3ccccc3[n+]2[H])CC1
T02
native IFP available
T02
selection_import_t02
0.864 1.000 0.612 native_similarity final_rank_score -26.0159 -0.781742 18 2 Pose
Z1820095916
[H]N(Cc1cccs1)C(=O)C1CCN(c2n(Cc3cc(C)ccc3C)c3ccccc3[n+]2[H])CC1
T01
native IFP available
T01
selection_import_t01
0.844 1.000 0.555 native_similarity final_rank_score -26.7758 -0.831354 19 1 Pose
Z1820095916
[H]N(Cc1cccs1)C(=O)C1CCN(c2n(Cc3cc(C)ccc3C)c3ccccc3[n+]2[H])CC1
T09
native IFP available
T09
selection_import_t09
0.823 1.000 0.493 native_similarity final_rank_score -23.4958 -0.775974 16 2 Pose
Z1820095916
[H]N(Cc1cccs1)C(=O)C1CCN(c2nc3ccccc3n2Cc2cc(C)ccc2C)CC1
T20
native IFP available
T20
selection_import_t20
0.812 1.000 0.463 native_similarity final_rank_score -41.0405 -0.590584 13 2 Pose
Z1820095916
[H]N(Cc1cccs1)C(=O)C1CCN(c2n(Cc3cc(C)ccc3C)c3ccccc3[n+]2[H])CC1
T03
native IFP available
T03
selection_import_t03
0.793 1.000 0.408 native_similarity final_rank_score -25.9677 -0.807099 15 2 Pose
Z1820095916
[H]N(Cc1cccs1)C(=O)C1CCN(c2n(Cc3cc(C)ccc3C)c3ccccc3[n+]2[H])CC1
T15
native IFP available
T15
selection_import_t15
0.793 1.000 0.408 native_similarity final_rank_score -26.0115 -0.763956 14 1 Pose
Z1820095916
[H]N(Cc1cccs1)C(=O)C1CCN(c2n(Cc3cc(C)ccc3C)c3ccccc3[n+]2[H])CC1
T18
native IFP available
T18
selection_import_t18
0.764 1.000 0.326 native_similarity final_rank_score -22.9985 -0.751494 11 3 Pose