FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 3 best compound-target hits listed 3 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T03T08T09
Z1551967334
[H][n+]1c(CCC)n(Cc2ccc(-c3ccccc3C(=O)O)cc2)c2cc(-c3nc4ccccc4n3C)cc(C)c21
0.853 0.843 2 0.85 0.83
Z1551967334
CCCc1nc2c(C)cc(-c3nc4ccccc4n3C)cc2n1Cc1ccc(-c2ccccc2C(=O)O)cc1
0.802 0.802 1 0.80

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z1551967334
[H][n+]1c(CCC)n(Cc2ccc(-c3ccccc3C(=O)O)cc2)c2cc(-c3nc4ccccc4n3C)cc(C)c21
T03
native IFP available
T03
selection_import_t03
0.853 1.000 0.579 native_similarity final_rank_score -29.8265 -0.690797 18 1 Pose
Z1551967334
[H][n+]1c(CCC)n(Cc2ccc(-c3ccccc3C(=O)O)cc2)c2cc(-c3nc4ccccc4n3C)cc(C)c21
T09
native IFP available
T09
selection_import_t09
0.834 1.000 0.526 native_similarity final_rank_score -30.6316 -0.679704 20 1 Pose
Z1551967334
CCCc1nc2c(C)cc(-c3nc4ccccc4n3C)cc2n1Cc1ccc(-c2ccccc2C(=O)O)cc1
T08
native IFP available
T08
selection_import_t08
0.802 1.000 0.434 native_similarity final_rank_score -32.9882 -0.821153 14 2 Pose