FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 3 best compound-target hits listed 3 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T03T15T17
OSA_Lib_85
[H][N+]1(CCC(=O)N2CC[C@]3([N+]4([H])CCCC4)C[C@H](c4ccccc4)[C@H]2[C@H](c2ccccc2)C3)CCN(C)CC1
0.874 0.874 1 0.87
OSA_Lib_85
[H][N+]1(C)CCN(CCC(=O)N2CC[C@]3([N+]4([H])CCCC4)C[C@H](c4ccccc4)[C@H]2[C@@H](c2ccccc2)C3)CC1
0.804 0.802 2 0.80 0.80

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OSA_Lib_85
[H][N+]1(CCC(=O)N2CC[C@]3([N+]4([H])CCCC4)C[C@H](c4ccccc4)[C@H]2[C@H](c2ccccc2)C3)CCN(C)CC1
T03
native IFP available
T03
selection_import_t03
0.874 1.000 0.639 native_similarity final_rank_score -23.6928 -0.723368 18 3 Pose
OSA_Lib_85
[H][N+]1(C)CCN(CCC(=O)N2CC[C@]3([N+]4([H])CCCC4)C[C@H](c4ccccc4)[C@H]2[C@@H](c2ccccc2)C3)CC1
T17
native IFP available
T17
selection_import_t17
0.804 1.000 0.440 native_similarity final_rank_score -20.6115 -0.603954 19 2 Pose
OSA_Lib_85
[H][N+]1(C)CCN(CCC(=O)N2CC[C@]3([N+]4([H])CCCC4)C[C@H](c4ccccc4)[C@H]2[C@@H](c2ccccc2)C3)CC1
T15
native IFP available
T15
selection_import_t15
0.801 1.000 0.431 native_similarity final_rank_score -23.1001 -0.64054 17 3 Pose