FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
Reset
3 compounds in matrix 3 best compound-target hits listed 3 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T11T15
OSA_Lib_241
[H][N+]1(CCCN2CC[C@]3([N+]4([H])CCCCC4)C[C@H](c4ccccc4)[C@H]2[C@@H](c2ccccc2)C3)CCCCC1
0.840 0.840 1 0.84
OSA_Lib_241
[H][N+]1(CCCN2CC[C@]3([N+]4([H])CCCCC4)C[C@@H](c4ccccc4)[C@H]2[C@H](c2ccccc2)C3)CCCCC1
0.830 0.830 1 0.83
OSA_Lib_241
[H][N+]1(CCC[N@+]2([H])CC[C@]3([N+]4([H])CCCCC4)C[C@H](c4ccccc4)[C@H]2[C@@H](c2ccccc2)C3)CCCCC1
0.793 0.793 1 0.79

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OSA_Lib_241
[H][N+]1(CCCN2CC[C@]3([N+]4([H])CCCCC4)C[C@H](c4ccccc4)[C@H]2[C@@H](c2ccccc2)C3)CCCCC1
T11
native IFP available
T11
selection_import_t11
0.840 1.000 0.542 native_similarity final_rank_score -22.7071 -0.669135 15 1 Pose
OSA_Lib_241
[H][N+]1(CCCN2CC[C@]3([N+]4([H])CCCCC4)C[C@@H](c4ccccc4)[C@H]2[C@H](c2ccccc2)C3)CCCCC1
T01
native IFP available
T01
selection_import_t01
0.830 1.000 0.515 native_similarity final_rank_score -22.3227 -0.714359 21 0 Pose
OSA_Lib_241
[H][N+]1(CCC[N@+]2([H])CC[C@]3([N+]4([H])CCCCC4)C[C@H](c4ccccc4)[C@H]2[C@@H](c2ccccc2)C3)CCCCC1
T15
native IFP available
T15
selection_import_t15
0.793 1.000 0.408 native_similarity final_rank_score -22.479 -0.694403 14 2 Pose