FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
Reset
2 compounds in matrix 2 best compound-target hits listed 2 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02
OHD_TB2022_11
[H]N([H])c1nc(N2CCN(C(=O)Cc3ccc(OCc4ccccc4)cc3)CC2)nc2cc(OC)c(OC)cc12
0.809 0.809 1 0.81
OHD_TB2022_11
[H]N([H])c1c2cc(OC)c(OC)cc2nc(N2CCN(C(=O)Cc3ccc(OCc4ccccc4)cc3)CC2)[n+]1[H]
0.809 0.809 1 0.81

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OHD_TB2022_11
[H]N([H])c1nc(N2CCN(C(=O)Cc3ccc(OCc4ccccc4)cc3)CC2)nc2cc(OC)c(OC)cc12
T01
native IFP available
T01
selection_import_t01
0.809 1.000 0.454 native_similarity final_rank_score -24.6624 -0.710656 19 2 Pose
OHD_TB2022_11
[H]N([H])c1c2cc(OC)c(OC)cc2nc(N2CCN(C(=O)Cc3ccc(OCc4ccccc4)cc3)CC2)[n+]1[H]
T02
native IFP available
T02
selection_import_t02
0.809 1.000 0.454 native_similarity final_rank_score -21.6229 -0.701776 19 2 Pose