FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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1 compounds in matrix 13 best compound-target hits listed 13 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T04T05T08T09T11T12T13T14T16T17T18
OHD_MAC_46
[H]Oc1cc(/C=N/Nc2ncnc3c(N([H])c4cccnc4)ncnc23)ccc1O
0.911 0.825 13 0.84 0.83 0.87 0.81 0.81 0.80 0.86 0.91 0.88 0.79 0.82 0.74 0.76

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OHD_MAC_46
[H]Oc1cc(/C=N/Nc2ncnc3c(N([H])c4cccnc4)ncnc23)ccc1O
T12
native IFP available
T12
selection_import_t12
0.911 1.000 0.745 native_similarity final_rank_score -26.7944 -1.07371 17 13 Pose
OHD_MAC_46
[H]Oc1cc(/C=N/Nc2ncnc3c(N([H])c4cccnc4)ncnc23)ccc1O
T13
native IFP available
T13
selection_import_t13
0.885 1.000 0.670 native_similarity final_rank_score -29.739 -1.12345 23 14 Pose
OHD_MAC_46
[H]Oc1cc(/C=N/Nc2ncnc3c(N([H])c4cccnc4)ncnc23)ccc1O
T04
native IFP available
T04
selection_import_t04
0.874 1.000 0.639 native_similarity final_rank_score -22.7368 -0.859654 13 8 Pose
OHD_MAC_46
[H]Oc1cc(/C=N/Nc2ncnc3c(N([H])c4cccnc4)ncnc23)ccc1O
T11
native IFP available
T11
selection_import_t11
0.862 1.000 0.607 native_similarity final_rank_score -23.4774 -0.942434 19 6 Pose
OHD_MAC_46
[H]Oc1cc(/C=N/Nc2ncnc3c(N([H])c4cccnc4)ncnc23)ccc1O
T01
native IFP available
T01
selection_import_t01
0.838 1.000 0.536 native_similarity final_rank_score -19.0807 -0.967321 17 7 Pose
OHD_MAC_46
[H]Oc1cc(/C=N/Nc2ncnc3c(N([H])c4cccnc4)ncnc23)ccc1O
T02
native IFP available
T02
selection_import_t02
0.832 1.000 0.519 native_similarity final_rank_score -25.4644 -0.936048 17 5 Pose
OHD_MAC_46
[H]Oc1cc(/C=N/Nc2ncnc3c(N([H])c4cccnc4)ncnc23)ccc1O
T16
native IFP available
T16
selection_import_t16
0.815 1.000 0.472 native_similarity final_rank_score -16.8076 -0.815812 16 5 Pose
OHD_MAC_46
[H]Oc1cc(/C=N/Nc2ncnc3c(N([H])c4cccnc4)ncnc23)ccc1O
T05
native IFP available
T05
selection_import_t05
0.813 1.000 0.465 native_similarity final_rank_score -27.3797 -1.11493 15 8 Pose
OHD_MAC_46
[H]Oc1cc(/C=N/Nc2ncnc3c(N([H])c4cccnc4)ncnc23)ccc1O
T08
native IFP available
T08
selection_import_t08
0.806 1.000 0.445 native_similarity final_rank_score -35.2625 -1.34752 15 10 Pose
OHD_MAC_46
[H]Oc1cc(/C=N/Nc2ncnc3c(N([H])c4cccnc4)ncnc23)ccc1O
T09
native IFP available
T09
selection_import_t09
0.802 1.000 0.433 native_similarity final_rank_score -25.148 -1.11347 15 7 Pose
OHD_MAC_46
[H]Oc1cc(/C=N/Nc2ncnc3c(N([H])c4cccnc4)ncnc23)ccc1O
T14
native IFP available
T14
selection_import_t14
0.794 1.000 0.411 native_similarity final_rank_score -21.7673 -0.88846 15 7 Pose
OHD_MAC_46
[H]Oc1cc(/C=N/Nc2ncnc3c(N([H])c4cccnc4)ncnc23)ccc1O
T18
native IFP available
T18
selection_import_t18
0.758 1.000 0.309 native_similarity final_rank_score -21.7204 -0.743151 13 8 Pose
OHD_MAC_46
[H]Oc1cc(/C=N/Nc2ncnc3c(N([H])c4cccnc4)ncnc23)ccc1O
T17
native IFP available
T17
selection_import_t17
0.736 1.000 0.246 native_similarity final_rank_score -22.757 -0.900748 19 8 Pose