FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 7 best compound-target hits listed 7 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T10T13T17T18T19T20
OHD_MAC_31
[H]Oc1ccc(/C=[N+]([H])/N=c2\ncn([H])c3c(N([H])c4ccc(F)c(Cl)c4)[n+]([H])cnc23)cc1OC
0.944 0.881 3 0.94 0.77 0.93
OHD_MAC_31
[H]Oc1ccc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(F)c(Cl)c4)ncnc23)cc1OC
0.881 0.811 4 0.86 0.88 0.76 0.75

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OHD_MAC_31
[H]Oc1ccc(/C=[N+]([H])/N=c2\ncn([H])c3c(N([H])c4ccc(F)c(Cl)c4)[n+]([H])cnc23)cc1OC
T10
native IFP available
T10
selection_import_t10
0.944 1.000 0.841 native_similarity final_rank_score -18.6428 -0.886465 18 10 Pose
OHD_MAC_31
[H]Oc1ccc(/C=[N+]([H])/N=c2\ncn([H])c3c(N([H])c4ccc(F)c(Cl)c4)[n+]([H])cnc23)cc1OC
T20
native IFP available
T20
selection_import_t20
0.929 1.000 0.796 native_similarity final_rank_score -15.1218 -0.627915 11 7 Pose
OHD_MAC_31
[H]Oc1ccc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(F)c(Cl)c4)ncnc23)cc1OC
T13
native IFP available
T13
selection_import_t13
0.881 1.000 0.661 native_similarity final_rank_score -30.3453 -1.06008 24 14 Pose
OHD_MAC_31
[H]Oc1ccc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(F)c(Cl)c4)ncnc23)cc1OC
T02
native IFP available
T02
selection_import_t02
0.859 1.000 0.599 native_similarity final_rank_score -22.6528 -0.853089 19 3 Pose
OHD_MAC_31
[H]Oc1ccc(/C=[N+]([H])/N=c2\ncn([H])c3c(N([H])c4ccc(F)c(Cl)c4)[n+]([H])cnc23)cc1OC
T17
native IFP available
T17
selection_import_t17
0.769 1.000 0.339 native_similarity final_rank_score -18.2217 -0.725305 19 5 Pose
OHD_MAC_31
[H]Oc1ccc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(F)c(Cl)c4)ncnc23)cc1OC
T18
native IFP available
T18
selection_import_t18
0.758 1.000 0.309 native_similarity final_rank_score -21.1554 -0.675533 13 7 Pose
OHD_MAC_31
[H]Oc1ccc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(F)c(Cl)c4)ncnc23)cc1OC
T19
native IFP available
T19
selection_import_t19
0.745 1.000 0.272 native_similarity final_rank_score -25.4797 -1.06308 22 9 Pose