FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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1 compounds in matrix 13 best compound-target hits listed 13 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T03T05T08T09T13T15T17T18T20T21T22
OHD_Leishmania_481
[H]Oc1cccc(/C=C/C(=N\N([H])C(=S)N([H])[H])c2cccc(N([H])C(=O)N([H])c3ccc(Cl)cc3)c2)c1
0.953 0.845 13 0.83 0.85 0.79 0.86 0.84 0.79 0.88 0.82 0.89 0.78 0.95 0.86 0.83

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OHD_Leishmania_481
[H]Oc1cccc(/C=C/C(=N\N([H])C(=S)N([H])[H])c2cccc(N([H])C(=O)N([H])c3ccc(Cl)cc3)c2)c1
T20
native IFP available
T20
selection_import_t20
0.953 1.000 0.867 native_similarity final_rank_score -24.0235 -0.708066 12 9 Pose
OHD_Leishmania_481
[H]Oc1cccc(/C=C/C(=N\N([H])C(=S)N([H])[H])c2cccc(N([H])C(=O)N([H])c3ccc(Cl)cc3)c2)c1
T17
native IFP available
T17
selection_import_t17
0.894 1.000 0.696 native_similarity final_rank_score -22.2153 -0.838847 18 6 Pose
OHD_Leishmania_481
[H]Oc1cccc(/C=C/C(=N\N([H])C(=S)N([H])[H])c2cccc(N([H])C(=O)N([H])c3ccc(Cl)cc3)c2)c1
T13
native IFP available
T13
selection_import_t13
0.885 1.000 0.670 native_similarity final_rank_score -19.7644 -1.00267 23 8 Pose
OHD_Leishmania_481
[H]Oc1cccc(/C=C/C(=N\N([H])C(=S)N([H])[H])c2cccc(N([H])C(=O)N([H])c3ccc(Cl)cc3)c2)c1
T21
native IFP available
T21
selection_import_t21
0.857 1.000 0.592 native_similarity final_rank_score -15.2577 -0.781504 17 9 Pose
OHD_Leishmania_481
[H]Oc1cccc(/C=C/C(=N\N([H])C(=S)N([H])[H])c2cccc(N([H])C(=O)N([H])c3ccc(Cl)cc3)c2)c1
T05
native IFP available
T05
selection_import_t05
0.856 1.000 0.590 native_similarity final_rank_score -26.4163 -1.04112 17 8 Pose
OHD_Leishmania_481
[H]Oc1cccc(/C=C/C(=N\N([H])C(=S)N([H])[H])c2cccc(N([H])C(=O)N([H])c3ccc(Cl)cc3)c2)c1
T02
native IFP available
T02
selection_import_t02
0.851 1.000 0.574 native_similarity final_rank_score -24.6948 -0.8404 19 5 Pose
OHD_Leishmania_481
[H]Oc1cccc(/C=C/C(=N\N([H])C(=S)N([H])[H])c2cccc(N([H])C(=O)N([H])c3ccc(Cl)cc3)c2)c1
T08
native IFP available
T08
selection_import_t08
0.844 1.000 0.556 native_similarity final_rank_score -25.2363 -1.05679 17 11 Pose
OHD_Leishmania_481
[H]Oc1cccc(/C=C/C(=N\N([H])C(=S)N([H])[H])c2cccc(N([H])C(=O)N([H])c3ccc(Cl)cc3)c2)c1
T01
native IFP available
T01
selection_import_t01
0.830 1.000 0.514 native_similarity final_rank_score -24.4886 -0.816536 19 6 Pose
OHD_Leishmania_481
[H]Oc1cccc(/C=C/C(=N\N([H])C(=S)N([H])[H])c2cccc(N([H])C(=O)N([H])c3ccc(Cl)cc3)c2)c1
T22
native IFP available
T22
selection_import_t22
0.829 1.000 0.512 native_similarity final_rank_score -27.8948 -0.951446 20 5 Pose
OHD_Leishmania_481
[H]Oc1cccc(/C=C/C(=N\N([H])C(=S)N([H])[H])c2cccc(N([H])C(=O)N([H])c3ccc(Cl)cc3)c2)c1
T15
native IFP available
T15
selection_import_t15
0.820 1.000 0.485 native_similarity final_rank_score -22.2054 -0.858902 17 6 Pose
OHD_Leishmania_481
[H]Oc1cccc(/C=C/C(=N\N([H])C(=S)N([H])[H])c2cccc(N([H])C(=O)N([H])c3ccc(Cl)cc3)c2)c1
T09
native IFP available
T09
selection_import_t09
0.794 1.000 0.412 native_similarity final_rank_score -26.2704 -0.854228 15 5 Pose
OHD_Leishmania_481
[H]Oc1cccc(/C=C/C(=N\N([H])C(=S)N([H])[H])c2cccc(N([H])C(=O)N([H])c3ccc(Cl)cc3)c2)c1
T03
native IFP available
T03
selection_import_t03
0.793 1.000 0.408 native_similarity final_rank_score -24.7699 -0.8945 15 4 Pose
OHD_Leishmania_481
[H]Oc1cccc(/C=C/C(=N\N([H])C(=S)N([H])[H])c2cccc(N([H])C(=O)N([H])c3ccc(Cl)cc3)c2)c1
T18
native IFP available
T18
selection_import_t18
0.785 1.000 0.385 native_similarity final_rank_score -23.0094 -0.787662 11 6 Pose