FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 7 best compound-target hits listed 7 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T04T08T17T20T21
OHD_Leishmania_356
[H]O[C@@H](COc1cc(=O)oc2ccccc12)CN1C(=O)/C(=N\N([H])C(=O)c2ccncc2)c2ccccc21
0.922 0.878 2 0.83 0.92
OHD_Leishmania_356
[H]O[C@H](COc1cc(=O)oc2ccccc12)CN1C(=O)/C(=N\N([H])C(=O)c2ccncc2)c2ccccc21
0.916 0.869 5 0.86 0.86 0.82 0.92 0.90

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OHD_Leishmania_356
[H]O[C@@H](COc1cc(=O)oc2ccccc12)CN1C(=O)/C(=N\N([H])C(=O)c2ccncc2)c2ccccc21
T20
native IFP available
T20
selection_import_t20
0.922 1.000 0.778 native_similarity final_rank_score -10.5927 -0.562159 12 7 Pose
OHD_Leishmania_356
[H]O[C@H](COc1cc(=O)oc2ccccc12)CN1C(=O)/C(=N\N([H])C(=O)c2ccncc2)c2ccccc21
T17
native IFP available
T17
selection_import_t17
0.916 1.000 0.761 native_similarity final_rank_score -17.5086 -0.618121 17 4 Pose
OHD_Leishmania_356
[H]O[C@H](COc1cc(=O)oc2ccccc12)CN1C(=O)/C(=N\N([H])C(=O)c2ccncc2)c2ccccc21
T21
native IFP available
T21
selection_import_t21
0.897 1.000 0.705 native_similarity final_rank_score -21.8866 -0.762846 18 13 Pose
OHD_Leishmania_356
[H]O[C@H](COc1cc(=O)oc2ccccc12)CN1C(=O)/C(=N\N([H])C(=O)c2ccncc2)c2ccccc21
T01
native IFP available
T01
selection_import_t01
0.855 1.000 0.586 native_similarity final_rank_score -24.971 -0.772957 20 3 Pose
OHD_Leishmania_356
[H]O[C@H](COc1cc(=O)oc2ccccc12)CN1C(=O)/C(=N\N([H])C(=O)c2ccncc2)c2ccccc21
T02
native IFP available
T02
selection_import_t02
0.855 1.000 0.586 native_similarity final_rank_score -26.1341 -0.804232 20 3 Pose
OHD_Leishmania_356
[H]O[C@@H](COc1cc(=O)oc2ccccc12)CN1C(=O)/C(=N\N([H])C(=O)c2ccncc2)c2ccccc21
T04
native IFP available
T04
selection_import_t04
0.834 1.000 0.525 native_similarity final_rank_score -19.6428 -0.724132 11 3 Pose
OHD_Leishmania_356
[H]O[C@H](COc1cc(=O)oc2ccccc12)CN1C(=O)/C(=N\N([H])C(=O)c2ccncc2)c2ccccc21
T08
native IFP available
T08
selection_import_t08
0.824 1.000 0.497 native_similarity final_rank_score -29.4576 -0.942471 16 7 Pose