FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 6 best compound-target hits listed 6 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T12T14T16T20T22
OHD_Babesia_16
[H]Oc1c2c(c(O[H])c3c1C(=O)c1ccccc1C3=O)[C@@H](O[C@H]1C[C@H]([N+]([H])([H])[H])[C@H](O[H])[C@H](C)O1)C[C@](O[H])(C(C)=O)C2
0.917 0.827 4 0.84 0.78 0.76 0.92
OHD_Babesia_16
[H]Oc1c2c(c(O[H])c3c1C(=O)c1ccccc1C3=O)[C@@H](O[C@H]1C[C@H](N([H])[H])[C@H](O[H])[C@H](C)O1)C[C@](O[H])(C(C)=O)C2
0.901 0.878 2 0.90 0.86

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OHD_Babesia_16
[H]Oc1c2c(c(O[H])c3c1C(=O)c1ccccc1C3=O)[C@@H](O[C@H]1C[C@H]([N+]([H])([H])[H])[C@H](O[H])[C@H](C)O1)C[C@](O[H])(C(C)=O)C2
T20
native IFP available
T20
selection_import_t20
0.917 1.000 0.763 native_similarity final_rank_score -26.9022 -0.755699 13 8 Pose
OHD_Babesia_16
[H]Oc1c2c(c(O[H])c3c1C(=O)c1ccccc1C3=O)[C@@H](O[C@H]1C[C@H](N([H])[H])[C@H](O[H])[C@H](C)O1)C[C@](O[H])(C(C)=O)C2
T12
native IFP available
T12
selection_import_t12
0.901 1.000 0.717 native_similarity final_rank_score -31.6917 -0.91144 20 12 Pose
OHD_Babesia_16
[H]Oc1c2c(c(O[H])c3c1C(=O)c1ccccc1C3=O)[C@@H](O[C@H]1C[C@H](N([H])[H])[C@H](O[H])[C@H](C)O1)C[C@](O[H])(C(C)=O)C2
T22
native IFP available
T22
selection_import_t22
0.856 1.000 0.588 native_similarity final_rank_score -32.8827 -0.934999 21 8 Pose
OHD_Babesia_16
[H]Oc1c2c(c(O[H])c3c1C(=O)c1ccccc1C3=O)[C@@H](O[C@H]1C[C@H]([N+]([H])([H])[H])[C@H](O[H])[C@H](C)O1)C[C@](O[H])(C(C)=O)C2
T02
native IFP available
T02
selection_import_t02
0.844 1.000 0.555 native_similarity final_rank_score -27.3156 -0.70587 19 6 Pose
OHD_Babesia_16
[H]Oc1c2c(c(O[H])c3c1C(=O)c1ccccc1C3=O)[C@@H](O[C@H]1C[C@H]([N+]([H])([H])[H])[C@H](O[H])[C@H](C)O1)C[C@](O[H])(C(C)=O)C2
T14
native IFP available
T14
selection_import_t14
0.784 1.000 0.382 native_similarity final_rank_score -25.4339 -0.681665 15 9 Pose
OHD_Babesia_16
[H]Oc1c2c(c(O[H])c3c1C(=O)c1ccccc1C3=O)[C@@H](O[C@H]1C[C@H]([N+]([H])([H])[H])[C@H](O[H])[C@H](C)O1)C[C@](O[H])(C(C)=O)C2
T16
native IFP available
T16
selection_import_t16
0.763 1.000 0.322 native_similarity final_rank_score -26.2231 -0.654866 14 4 Pose