FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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1 compounds in matrix 9 best compound-target hits listed 9 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T03T06T10T14T15T16T22
NMT-TY0565
[H]N([H])c1ccc(S(=O)(=O)N([H])c2c(O)ncnc2N([H])[H])cc1
0.884 0.820 9 0.85 0.85 0.84 0.88 0.85 0.78 0.77 0.76 0.79

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
NMT-TY0565
[H]N([H])c1ccc(S(=O)(=O)N([H])c2c(O)ncnc2N([H])[H])cc1
T06
native IFP available
T06
selection_import_t06
0.884 1.000 0.669 native_similarity final_rank_score -22.9835 -1.3133 17 5 Pose
NMT-TY0565
[H]N([H])c1ccc(S(=O)(=O)N([H])c2c(O)ncnc2N([H])[H])cc1
T02
native IFP available
T02
selection_import_t02
0.853 1.000 0.580 native_similarity final_rank_score -25.8069 -1.42184 14 7 Pose
NMT-TY0565
[H]N([H])c1ccc(S(=O)(=O)N([H])c2c(O)ncnc2N([H])[H])cc1
T01
native IFP available
T01
selection_import_t01
0.851 1.000 0.573 native_similarity final_rank_score -25.9702 -1.42538 15 8 Pose
NMT-TY0565
[H]N([H])c1ccc(S(=O)(=O)N([H])c2c(O)ncnc2N([H])[H])cc1
T10
native IFP available
T10
selection_import_t10
0.849 1.000 0.569 native_similarity final_rank_score -25.553 -1.35686 13 12 Pose
NMT-TY0565
[H]N([H])c1ccc(S(=O)(=O)N([H])c2c(O)ncnc2N([H])[H])cc1
T03
native IFP available
T03
selection_import_t03
0.843 1.000 0.550 native_similarity final_rank_score -26.5605 -1.52753 15 10 Pose
NMT-TY0565
[H]N([H])c1ccc(S(=O)(=O)N([H])c2c(O)ncnc2N([H])[H])cc1
T22
native IFP available
T22
selection_import_t22
0.790 1.000 0.400 native_similarity final_rank_score -30.7231 -1.67804 19 16 Pose
NMT-TY0565
[H]N([H])c1ccc(S(=O)(=O)N([H])c2c(O)ncnc2N([H])[H])cc1
T14
native IFP available
T14
selection_import_t14
0.778 1.000 0.366 native_similarity final_rank_score -21.6592 -1.16101 10 8 Pose
NMT-TY0565
[H]N([H])c1ccc(S(=O)(=O)N([H])c2c(O)ncnc2N([H])[H])cc1
T15
native IFP available
T15
selection_import_t15
0.774 1.000 0.353 native_similarity final_rank_score -23.0227 -1.28783 14 9 Pose
NMT-TY0565
[H]N([H])c1ccc(S(=O)(=O)N([H])c2c(O)ncnc2N([H])[H])cc1
T16
native IFP available
T16
selection_import_t16
0.763 1.000 0.322 native_similarity final_rank_score -23.2122 -1.28108 14 8 Pose