FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T12T19T20T22
KB_chagas_26
[H]N([C@H]1CC[C@@H](Oc2cc3cnccc3cc2-c2ccsc2)CC1)S(C)(=O)=O
0.932 0.829 2 0.93 0.73
KB_chagas_26
[H]N([C@H]1CC[C@@H](Oc2cc3c[n+]([H])ccc3cc2-c2ccsc2)CC1)S(C)(=O)=O
0.914 0.865 2 0.82 0.91

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
KB_chagas_26
[H]N([C@H]1CC[C@@H](Oc2cc3cnccc3cc2-c2ccsc2)CC1)S(C)(=O)=O
T12
native IFP available
T12
selection_import_t12
0.932 1.000 0.807 native_similarity final_rank_score -27.2417 -1.05988 19 11 Pose
KB_chagas_26
[H]N([C@H]1CC[C@@H](Oc2cc3c[n+]([H])ccc3cc2-c2ccsc2)CC1)S(C)(=O)=O
T22
native IFP available
T22
selection_import_t22
0.914 1.000 0.753 native_similarity final_rank_score -26.5244 -1.25727 20 8 Pose
KB_chagas_26
[H]N([C@H]1CC[C@@H](Oc2cc3c[n+]([H])ccc3cc2-c2ccsc2)CC1)S(C)(=O)=O
T20
native IFP available
T20
selection_import_t20
0.817 1.000 0.478 native_similarity final_rank_score -22.7101 -0.79544 12 5 Pose
KB_chagas_26
[H]N([C@H]1CC[C@@H](Oc2cc3cnccc3cc2-c2ccsc2)CC1)S(C)(=O)=O
T19
native IFP available
T19
selection_import_t19
0.725 1.000 0.215 native_similarity final_rank_score -34.6324 -1.32575 19 8 Pose