FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 7 best compound-target hits listed 7 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T03T08T09T17T20
KB_HAT_67
[H][n+]1ccc(N2CCN(C(=O)c3cccc(-c4cccnc4)c3)CC2)nc1N(C)[C@H]1CC[N@+]([H])(C)CC1
0.904 0.838 6 0.85 0.85 0.82 0.82 0.77 0.90
KB_HAT_67
[H][N@+]1(C)CC[C@H](N(C)c2nccc(N3CCN(C(=O)c4cccc(-c5cccnc5)c4)CC3)n2)CC1
0.812 0.812 1 0.81

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
KB_HAT_67
[H][n+]1ccc(N2CCN(C(=O)c3cccc(-c4cccnc4)c3)CC2)nc1N(C)[C@H]1CC[N@+]([H])(C)CC1
T20
native IFP available
T20
selection_import_t20
0.904 1.000 0.725 native_similarity final_rank_score -22.4332 -0.545176 10 2 Pose
KB_HAT_67
[H][n+]1ccc(N2CCN(C(=O)c3cccc(-c4cccnc4)c3)CC2)nc1N(C)[C@H]1CC[N@+]([H])(C)CC1
T02
native IFP available
T02
selection_import_t02
0.855 1.000 0.584 native_similarity final_rank_score -25.367 -0.76336 18 2 Pose
KB_HAT_67
[H][n+]1ccc(N2CCN(C(=O)c3cccc(-c4cccnc4)c3)CC2)nc1N(C)[C@H]1CC[N@+]([H])(C)CC1
T01
native IFP available
T01
selection_import_t01
0.851 1.000 0.574 native_similarity final_rank_score -28.9895 -0.786359 19 3 Pose
KB_HAT_67
[H][n+]1ccc(N2CCN(C(=O)c3cccc(-c4cccnc4)c3)CC2)nc1N(C)[C@H]1CC[N@+]([H])(C)CC1
T03
native IFP available
T03
selection_import_t03
0.822 1.000 0.491 native_similarity final_rank_score -26.8363 -0.832458 15 3 Pose
KB_HAT_67
[H][n+]1ccc(N2CCN(C(=O)c3cccc(-c4cccnc4)c3)CC2)nc1N(C)[C@H]1CC[N@+]([H])(C)CC1
T08
native IFP available
T08
selection_import_t08
0.822 1.000 0.491 native_similarity final_rank_score -30.8274 -0.97212 17 2 Pose
KB_HAT_67
[H][N@+]1(C)CC[C@H](N(C)c2nccc(N3CCN(C(=O)c4cccc(-c5cccnc5)c4)CC3)n2)CC1
T09
native IFP available
T09
selection_import_t09
0.812 1.000 0.464 native_similarity final_rank_score -30.8426 -0.792379 18 1 Pose
KB_HAT_67
[H][n+]1ccc(N2CCN(C(=O)c3cccc(-c4cccnc4)c3)CC2)nc1N(C)[C@H]1CC[N@+]([H])(C)CC1
T17
native IFP available
T17
selection_import_t17
0.773 1.000 0.352 native_similarity final_rank_score -24.6203 -0.6505 17 3 Pose