FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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3 compounds in matrix 6 best compound-target hits listed 6 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T09T14T16T17T18T20
Z56958950
[H]N(C(=O)CN1C(=O)/C(=C2/SC(=S)N([C@@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccc(OC)cc1
0.912 0.853 2 0.91 0.79
Z56958950
[H]N(C(=O)CN1C(=O)/C(=C2\SC(=S)N([C@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccc(OC)cc1
0.815 0.805 2 0.79 0.82
Z56958950
[H]N(C(=O)CN1C(=O)/C(=C2\SC(=S)N([C@@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccc(OC)cc1
0.789 0.775 2 0.79 0.76

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z56958950
[H]N(C(=O)CN1C(=O)/C(=C2/SC(=S)N([C@@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccc(OC)cc1
T09
native IFP available
T09
selection_import_t09
0.912 1.000 0.749 native_similarity final_rank_score -27.8666 -0.775488 21 4 Pose
Z56958950
[H]N(C(=O)CN1C(=O)/C(=C2\SC(=S)N([C@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccc(OC)cc1
T16
native IFP available
T16
selection_import_t16
0.815 1.000 0.472 native_similarity final_rank_score -21.3015 -0.63054 16 2 Pose
Z56958950
[H]N(C(=O)CN1C(=O)/C(=C2\SC(=S)N([C@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccc(OC)cc1
T14
native IFP available
T14
selection_import_t14
0.795 1.000 0.413 native_similarity final_rank_score -17.4659 -0.616701 17 6 Pose
Z56958950
[H]N(C(=O)CN1C(=O)/C(=C2/SC(=S)N([C@@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccc(OC)cc1
T20
native IFP available
T20
selection_import_t20
0.793 1.000 0.410 native_similarity final_rank_score -13.5563 -0.536855 11 6 Pose
Z56958950
[H]N(C(=O)CN1C(=O)/C(=C2\SC(=S)N([C@@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccc(OC)cc1
T17
native IFP available
T17
selection_import_t17
0.789 1.000 0.396 native_similarity final_rank_score -22.9231 -0.643045 18 2 Pose
Z56958950
[H]N(C(=O)CN1C(=O)/C(=C2\SC(=S)N([C@@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccc(OC)cc1
T18
native IFP available
T18
selection_import_t18
0.761 1.000 0.317 native_similarity final_rank_score -21.175 -0.605114 12 3 Pose