FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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2 compounds in matrix 11 best compound-target hits listed 11 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T03T04T05T07T08T09T11T12T15
OHD_TB2022_21
[H]N([H])c1nc(N([H])[H])[n+]([H])c2ncc(CN(Cc3ccccc3)Cc3ccc(Oc4ccc(OC)cc4)cc3)nc12
0.945 0.904 9 0.94 0.90 0.90 0.90 0.93 0.92 0.92 0.87 0.84
OHD_TB2022_21
[H]N([H])c1nc(N([H])[H])c2nc(CN(Cc3ccccc3)Cc3ccc(Oc4ccc(OC)cc4)cc3)cnc2n1
0.880 0.820 2 0.88 0.76

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OHD_TB2022_21
[H]N([H])c1nc(N([H])[H])[n+]([H])c2ncc(CN(Cc3ccccc3)Cc3ccc(Oc4ccc(OC)cc4)cc3)nc12
T01
native IFP available
T01
selection_import_t01
0.945 1.000 0.842 native_similarity final_rank_score -24.1835 -0.776562 21 11 Pose
OHD_TB2022_21
[H]N([H])c1nc(N([H])[H])[n+]([H])c2ncc(CN(Cc3ccccc3)Cc3ccc(Oc4ccc(OC)cc4)cc3)nc12
T07
native IFP available
T07
selection_import_t07
0.931 1.000 0.804 native_similarity final_rank_score -33.7036 -1.14596 21 7 Pose
OHD_TB2022_21
[H]N([H])c1nc(N([H])[H])[n+]([H])c2ncc(CN(Cc3ccccc3)Cc3ccc(Oc4ccc(OC)cc4)cc3)nc12
T08
native IFP available
T08
selection_import_t08
0.920 1.000 0.771 native_similarity final_rank_score -33.4245 -1.14683 20 7 Pose
OHD_TB2022_21
[H]N([H])c1nc(N([H])[H])[n+]([H])c2ncc(CN(Cc3ccccc3)Cc3ccc(Oc4ccc(OC)cc4)cc3)nc12
T11
native IFP available
T11
selection_import_t11
0.916 1.000 0.761 native_similarity final_rank_score -23.6267 -0.711971 16 8 Pose
OHD_TB2022_21
[H]N([H])c1nc(N([H])[H])[n+]([H])c2ncc(CN(Cc3ccccc3)Cc3ccc(Oc4ccc(OC)cc4)cc3)nc12
T05
native IFP available
T05
selection_import_t05
0.904 1.000 0.727 native_similarity final_rank_score -24.9697 -0.785109 18 4 Pose
OHD_TB2022_21
[H]N([H])c1nc(N([H])[H])[n+]([H])c2ncc(CN(Cc3ccccc3)Cc3ccc(Oc4ccc(OC)cc4)cc3)nc12
T02
native IFP available
T02
selection_import_t02
0.904 1.000 0.726 native_similarity final_rank_score -22.3917 -0.734977 24 9 Pose
OHD_TB2022_21
[H]N([H])c1nc(N([H])[H])[n+]([H])c2ncc(CN(Cc3ccccc3)Cc3ccc(Oc4ccc(OC)cc4)cc3)nc12
T03
native IFP available
T03
selection_import_t03
0.901 1.000 0.718 native_similarity final_rank_score -29.7543 -0.965604 21 10 Pose
OHD_TB2022_21
[H]N([H])c1nc(N([H])[H])c2nc(CN(Cc3ccccc3)Cc3ccc(Oc4ccc(OC)cc4)cc3)cnc2n1
T04
native IFP available
T04
selection_import_t04
0.880 1.000 0.658 native_similarity final_rank_score -29.1901 -0.942905 14 6 Pose
OHD_TB2022_21
[H]N([H])c1nc(N([H])[H])[n+]([H])c2ncc(CN(Cc3ccccc3)Cc3ccc(Oc4ccc(OC)cc4)cc3)nc12
T12
native IFP available
T12
selection_import_t12
0.874 1.000 0.640 native_similarity final_rank_score -25.0202 -0.737164 19 11 Pose
OHD_TB2022_21
[H]N([H])c1nc(N([H])[H])[n+]([H])c2ncc(CN(Cc3ccccc3)Cc3ccc(Oc4ccc(OC)cc4)cc3)nc12
T15
native IFP available
T15
selection_import_t15
0.842 1.000 0.548 native_similarity final_rank_score -22.2933 -0.717527 21 7 Pose
OHD_TB2022_21
[H]N([H])c1nc(N([H])[H])c2nc(CN(Cc3ccccc3)Cc3ccc(Oc4ccc(OC)cc4)cc3)cnc2n1
T09
native IFP available
T09
selection_import_t09
0.759 1.000 0.312 native_similarity final_rank_score -19.327 -0.68523 15 4 Pose