FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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2 compounds in matrix 3 best compound-target hits listed 2 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T10T17
MK14
[H]N(c1ccc(N2CCN(Cc3c4c(c(C)c(C)c3OC)OC(C)(C)CC4)CC2)cc1)S(C)(=O)=O
0.940 0.854 2 0.94 0.77
MK144
[H]OCc1cc(-c2ccc(O[H])cc2)no1
0.920 0.920 1 0.92

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
MK14
[H]N(c1ccc(N2CCN(Cc3c4c(c(C)c(C)c3OC)OC(C)(C)CC4)CC2)cc1)S(C)(=O)=O
T10
native IFP available
T10
selection_import_t10
0.940 1.000 0.829 native_similarity final_rank_score -25.848 -0.771667 17 11 Pose
MK144
[H]OCc1cc(-c2ccc(O[H])cc2)no1
T10
native IFP available
T10
selection_import_t10
0.920 1.000 0.772 native_similarity final_rank_score -19.0658 -1.73744 15 11 Pose
MK14
[H]N(c1ccc(N2CCN(Cc3c4c(c(C)c(C)c3OC)OC(C)(C)CC4)CC2)cc1)S(C)(=O)=O
T17
native IFP available
T17
selection_import_t17
0.769 1.000 0.339 native_similarity final_rank_score -22.8232 -0.668499 19 8 Pose